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- [1] Identification of novel series of human CCR1 antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (06) : 2215 - 2221Xie, Yun FengSircar, IlaLake, KirkKomandla, MallareddyLigsay, KathleenLi, JianXu, KuiParise, JasonSchneider, LisaHuang, DingqiuLiu, JupingSakurai, NaokiBarbosa, MiguelJack, Rick
- [2] MEDI 207-Discovery of novel, orally available piperidine-containing CCR1 antagonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232Lu, Shou-FuChou, Yuo-LingLee, WheeseongLiang, XiaolinPhillips, Gary B.Schlyer, SabineWei, Robert G.Xu, JinlouYu, HongyiGe, Xue SnowHarirchian, PaymannRibeiro, SofiaSubramanyam, BabuWalters, JanetteHoruk, RichardKochanny, Monica J.
- [3] MEDI 165-Discovery and optimization of a series of CCR4 antagonists from Hit to CDABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2008, 235Mete, AntonioAndrews, GlenBaxter, AndrewCheshire, DavidEwart, LornaHarper, SteveHickling, KevinKindon, NicholasMcGinnity, DermotMurray, ClaireStocks, MichaelTomkinson, NicholasWregget, KeithYoung, Simon
- [4] Novel, acidic CCR2 receptor antagonists: From hit to leadLETTERS IN DRUG DESIGN & DISCOVERY, 2007, 4 (03) : 185 - 191Zou, D.Zhai, H. A.Eckman, J.Higgins, P.Gillard, M.Knerr, L.Carre, S.Pasau, P.Collart, P.Grassi, J.Libertine, L.Nicolas, J. -M.Schwartz, C. E.
- [5] Discovery and Lead Optimization of a Novel Series of CC Chemokine Receptor 1 (CCR1)-Selective Piperidine Antagonists via Parallel SynthesisJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (22) : 9643 - 9653Cavallaro, Cullen L.Briceno, StephanieChen, JingCvijic, Mary EllenDavies, PaulHynes, John, Jr.Liu, Rui-QinMandlekar, SandhyaRose, Anne V.Tebben, Andrew J.Van Kirk, KatyWatson, AndrewWu, HongYang, GuchenCarter, Percy H.
- [6] From HTS hit to CD: Optimization of a novel series of CCR4 antagonistsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Mete, AntonioAndrews, GlenBaxter, AndrewCheshire, DavidEwart, LornaHarper, SteveHickling, KevinKindon, NicholasMcGinnity, DermotMurray, ClaireStocks, MichaelTomkinson, NicholasWregget, KeithYoung, Simon
- [7] The discovery of structurally novel CCR1 antagonists derived from a hydroxyethylene peptide isostere templateBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (09) : 2163 - 2167Kath, JCDiRico, APGladue, RPMartin, WHMcElroy, EBStock, IATylaska, LAZheng, DY
- [8] Discovery of ONO-7300243 from a Novel Class of Lysophosphatidic Acid Receptor 1 Antagonists: From Hit to LeadACS MEDICINAL CHEMISTRY LETTERS, 2016, 7 (10): : 913 - 918Terakado, MasahikoSuzuki, HidehiroHashimura, KazuyaTanaka, MotoyukiUeda, HideyukiKohno, HiroshiFujimoto, TakuSaga, HiroshiNakade, ShinjiHabashita, HiromuTakaoka, YoshikazuSeko, Takuya
- [9] Lead optimisation of the N1 substituent of a novel series of indazole arylsulfonamides as CCR4 antagonists and identification of a candidate for clinical investigationBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (08) : 2730 - 2733Procopiou, Panayiotis A.Ford, Alison J.Graves, Rebecca H.Hall, David A.Hodgson, Simon T.Lacroix, Yannick M. L.Needham, DeborahSlack, Robert J.