Design of potent and selective cathepsin K inhibitors which span the active site.

被引:0
作者
Thompson, SK
Halbert, SM
Michaud, E
Bossard, MJ
Tomaszek, TA
Levy, MA
Meek, TD
Zhao, B
Smith, WW
Janson, CA
McQueney, MS
AbdelMeguid, SS
Briand, J
Sarkar, SK
Huddleston, MJ
Ijames, CF
Carr, SA
DesJarlais, RL
Shu, A
Garnes, K
Heys, JR
Zembryki, D
LeeRykaczewski, LV
James, IE
Lark, M
Bradbeer, JN
Drake, FH
Gowen, M
Veber, DF
机构
[1] SMITHKLINE BEECHAM PHARMACEUT,DEPT MED CHEM,KING OF PRUSSIA,PA 19406
[2] SMITHKLINE BEECHAM PHARMACEUT,DEPT MOL RECOGNIT,KING OF PRUSSIA,PA 19406
[3] SMITHKLINE BEECHAM PHARMACEUT,DEPT MACROMOL SCI,KING OF PRUSSIA,PA 19406
[4] SMITHKLINE BEECHAM PHARMACEUT,DEPT PHYS & STRUCT CHEM,KING OF PRUSSIA,PA 19406
[5] SMITHKLINE BEECHAM PHARMACEUT,DEPT RADIOCHEM,KING OF PRUSSIA,PA 19406
[6] SMITHKLINE BEECHAM PHARMACEUT,DEPT CELLULAR BIOCHEM,KING OF PRUSSIA,PA 19406
来源
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 1997年 / 214卷
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D O I
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
引用
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页码:279 / MEDI
页数:1
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