Selective cyclooxygenase-2 inhibitors

被引:89
作者
Prasit, P
Riendeau, D
机构
[1] Merck Frosst Centre for Therapeutic Research, Pointe Claire-Dorval, Que. H9R 4P8
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 32 | 1997年 / 32卷
关键词
D O I
10.1016/S0065-7743(08)61479-7
中图分类号
O69 [应用化学];
学科分类号
081704 ;
摘要
[No abstract available]
引用
收藏
页码:211 / 220
页数:10
相关论文
共 81 条
[1]  
Adams J, 1996, J NEUROCHEM, V66, P6
[2]   PURIFICATION, CHARACTERIZATION AND SELECTIVE-INHIBITION OF HUMAN PROSTAGLANDIN-G/H SYNTHASE-1 AND SYNTHASE-2 EXPRESSED IN THE BACULOVIRUS SYSTEM [J].
BARNETT, J ;
CHOW, J ;
IVES, D ;
CHIOU, M ;
MACKENZIE, R ;
OSEN, E ;
NGUYEN, B ;
TSING, S ;
BACH, C ;
FREIRE, J ;
CHAN, H ;
SIGAL, E ;
RAMESHA, C .
BIOCHIMICA ET BIOPHYSICA ACTA-PROTEIN STRUCTURE AND MOLECULAR ENZYMOLOGY, 1994, 1209 (01) :130-139
[3]  
Barnett JW, Eur. Pat Appl., Patent No. [714895, EP 714895]
[4]  
BATT DG, Patent No. 9610012
[5]  
Bertenshaw S. R., [No title captured], Patent No. [WO 9515316, 9515316]
[6]  
BESWICK PJ, Patent No. 9631509
[7]  
BLACK C, Patent No. 9636623
[8]  
BLACK C, Patent No. 9619469
[9]   From indomethacin to a selective COX-2 inhibitor: Development of indolalkanoic acids as potent and selective cyclooxygenase-2 inhibitors [J].
Black, WC ;
Bayly, C ;
Belley, M ;
Chan, CC ;
Charleson, S ;
Denis, D ;
Gauthier, JY ;
Gordon, R ;
Guay, D ;
Kargman, S ;
Lau, CK ;
Leblanc, Y ;
Mancini, J ;
Ouellet, M ;
Percival, D ;
Roy, P ;
Skorey, K ;
Tagari, P ;
Vickers, P ;
Wong, E ;
Xu, L ;
Prasit, P .
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1996, 6 (06) :725-730
[10]   A human whole blood assay for clinical evaluation of biochemical efficacy of cyclooxygenase inhibitors [J].
Brideau, C ;
Kargman, S ;
Liu, S ;
Dallob, AL ;
Ehrich, EW ;
Rodger, IW ;
Chan, CC .
INFLAMMATION RESEARCH, 1996, 45 (02) :68-74