New routes to steroidal heterocyclic derivatives: Synthesis of biologically active pyrazolyl- and isoxazolylpregnene derivatives.

被引:14
作者
Abdelhamid, Abdou O. [1 ]
Abdelhalim, Mervat M.
Elmegeed, Gamall A.
机构
[1] Cairo Univ, Fac Sci, Dept Chem, Giza 12613, Egypt
[2] Natl Res Ctr, Hormone Dept, Giza 12622, Egypt
关键词
D O I
10.1002/jhet.5570440102
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Pyrazolyl- and isoxazolylpregnene derivatives were synthesized from the appropriate hydrazonoyl chlorides and hydroximoyl chlorides with enaminoprogesterone derivative. The newly synthesized compounds were elucidated by elemental analysis, spectral data and chemical transformation. Some products were tested towards some bacteria and some Fungal-plant pathogens.
引用
收藏
页码:7 / 11
页数:5
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