Facile synthesis of N-substituted pyrroles via microwave-induced bismuth nitrate-catalyzed reaction

被引：84

作者：

Rivera, Sonya ^{[1
]}

Bandyopadhyay, Debasish ^{[1
]}

Banik, Bimal K. ^{[1
]}

机构：

[1] Univ Texas Pan Amer, Dept Chem, Edinburg, TX 78539 USA

来源：

TETRAHEDRON LETTERS | 2009年 / 50卷 / 39期

关键词：

Pyrrole synthesis; Bismuth nitrate; Microwave irradiation; Polyaromatic compounds; POLYCYCLIC AROMATIC-COMPOUNDS; 1,3-DIPOLAR CYCLOADDITIONS; BIOLOGICAL EVALUATION; ANTICANCER AGENTS; BETA-LACTAMS; ENTRY;

D O I：

10.1016/j.tetlet.2009.06.002

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Simple synthesis of N-substituted pyrroles using microwave-induced bismuth nitrate-catalyzed reaction has been accomplished with an excellent yield. A plausible mechanism has been advanced. This reaction also provides a simple method to prepare diverse varieties of N-substituted pyrrole derivatives with less nucleophilic polyaromatic amines. (C) 2009 Published by Elsevier Ltd.

引用

页码：5445 / 5448

页数：4

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