BF3.OEt2-catalyzed one-pot three-component access to diarylmethylazides

被引：2
作者：
Prasad, Sure Siva
Joshi, Dirgha Raj
Kim, Ikyon [1 ]
机构：
[1] Yonsei Univ, Coll Pharm, 85 Songdogwahak Ro, Incheon 21983, South Korea
来源：
TETRAHEDRON LETTERS | 2021年 / 67卷
基金：
新加坡国家研究基金会;
关键词：
One-pot reaction; Multi-component reaction; Diarylmethylazide; Diversity-oriented synthesis;
D O I：
10.1016/j.tetlet.2020.152820
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A direct one-pot access to diarylmethylazides, versatile intermediates, from commercially available starting materials was enabled via three-component coupling of aldehydes, arenes, and TMSN3 in the presence of a catalytic amount of BF3.OEt2. (C) 2021 Elsevier Ltd. All rights reserved.
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页数：5
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