Rearrangement of 3,3-disubstituted indolenines and synthesis of 2,3-substituted indoles

被引：69

作者：

Liu, Kevin G. ^{[1
]}

Robichaud, Albert J. ^{[1
]}

Lo, Jennifer R. ^{[1
]}

Mattes, James F. ^{[1
]}

Cai, Yanxuan ^{[1
]}

机构：

[1] Wyeth Res, Chem & Screening Sci, Princeton, NJ 08543 USA

来源：

ORGANIC LETTERS | 2006年 / 8卷 / 25期

关键词：

D O I：

10.1021/ol0623567

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Synthesis of 2,3-substituted indoles from phenylhydrazine and alpha-branched aldehydes via rearrangement of 3,3-disubstituted indolenine intermediates is reported.

引用

页码：5769 / 5771

页数：3

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