Mild and efficient solvent-free Friedel-Crafts acylation of reserpine

被引：3
|
作者：
Begum, Sabira [1 ]
Zehra, Syeda Qamar [1 ]
Siddiqui, Bina S. [1 ]
机构：
[1] Univ Karachi, HEJ Res Inst Chem, Int Ctr Chem Sci, Karachi 75270, Pakistan
来源：
SYNTHETIC COMMUNICATIONS | 2006年 / 36卷 / 21期
关键词：
acyl reserpines; beta-carboline; Friedel-Crafts acylation; reserpine; solid-phase reaction;
D O I：
10.1080/00397910600908900
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The first mild, efficient, solvent-free Friedel - Crafts acylation of reserpine has been developed, which resulted in the synthesis of 10- and 12-acylated homologues in high overall yields.
引用
收藏
页码：3203 / 3224
页数：22
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