Mild and efficient solvent-free Friedel-Crafts acylation of reserpine

被引：3

作者：

Begum, Sabira ^{[1
]}

Zehra, Syeda Qamar ^{[1
]}

Siddiqui, Bina S. ^{[1
]}

机构：

[1] Univ Karachi, HEJ Res Inst Chem, Int Ctr Chem Sci, Karachi 75270, Pakistan

来源：

SYNTHETIC COMMUNICATIONS | 2006年 / 36卷 / 21期

关键词：

acyl reserpines; beta-carboline; Friedel-Crafts acylation; reserpine; solid-phase reaction;

D O I：

10.1080/00397910600908900

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The first mild, efficient, solvent-free Friedel - Crafts acylation of reserpine has been developed, which resulted in the synthesis of 10- and 12-acylated homologues in high overall yields.

引用

页码：3203 / 3224

页数：22

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