Synthesis of novel pyrazole-linked norcantharidin derivatives of substituted aromatic amines with efficient 1,3-dipolar cycloaddition

被引:4
作者
Deng, Liping [1 ]
Hu, Yongzhou [1 ]
机构
[1] Zhejiang Univ, Dept Med Chem, Sch Pharmaceut Sci, Hangzhou 310031, Peoples R China
关键词
D O I
10.1002/jhet.5570430646
中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
Highly efficient, practical and convient synthesis of fifteen compounds by the [3+2] 1,3-dipolar cycloaddition reaction of norcantharidin derivatives of substituted aromatic amines with three hydrazines in the presence of Chloramine-T.
引用
收藏
页码:1715 / 1719
页数:5
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