Synthesis of 4,5-disubstituted 1H-1,3,4,5-tetrahydrobenz[cd]indole derivatives

被引：0
作者：
Galambos, G
Csokasi, P
Szantay, C
Szantay, C
机构：
[1] CENT RES INST CHEM,H-1525 BUDAPEST,HUNGARY
[2] CHEM WORKS GEDEON RICHTER LTD,SPECT RES DEPT,H-1475 BUDAPEST,HUNGARY
来源：
LIEBIGS ANNALEN-RECUEIL | 1997年 / 09期
关键词：
3,4-disubstituted indoles; palladium-catalysed coupling; thio enol ether; radical addition; intramolecular cyclization;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Tetrahydrobenz[cd]indole derivatives (51-54) were synthesized from 4-iodo-3-(2'-nitroethyl)indole (10) via palladium-catalysed coupling with acetylenes followed by a thiol addition, an oxidation and an intramolecular Michael-addition.
引用
收藏
页码：1969 / 1978
页数：10
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