Dehydrogenative etherification homocoupling of heterocyclic N-oxides

被引：4

作者：

Zhang, Dong ^{[1
]}

Qiao, Kai ^{[1
]}

Yuan, Xin ^{[1
]}

Zheng, Mingwei ^{[1
]}

Fang, Zheng ^{[1
]}

Wan, Li ^{[1
,2
]}

Guo, Kai ^{[1
,2
]}

机构：

[1] Nanjing Tech Univ, Coll Biotechnol & Pharmaceut Engn, 30 Puzhu South Rd, Nanjing 211816, Jiangsu, Peoples R China

[2] Nanjing Tech Univ, State Key Lab Mat Oriented Chem Engn, 30 Puzhu South Rd, Nanjing 211816, Jiangsu, Peoples R China

来源：

TETRAHEDRON LETTERS | 2018年 / 59卷 / 18期

基金：

中国国家自然科学基金;

关键词：

Regioselective; Homocoupling; Quinoline; PyBroP; O-tethered; METAL-COMPLEXES; DNA; FUNCTIONALIZATION; RUTHENIUM(II); QUINOLINES; NITROGEN; LIGANDS; CARBON; CELLS; DRUG;

D O I：

10.1016/j.tetlet.2018.03.071

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A novel approach was developed for the dehydrogenative etherification homocoupling of heterocyclic N oxides in the presence of silver oxide and PyBroP. Various substrates were well tolerated and the desired products were obtained in moderate to good yields. Generally, this reaction features excellent functional group compatibility, broad substrate scope and good regioselectivity. (C) 2018 Elsevier Ltd. All rights reserved.

引用

收藏

页码：1752 / 1756

页数：5

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