Synthesis and Bio-Evaluation of Novel Salicylic Acid-Oriented Thiourea Derivatives with Potential Applications in Agriculture

被引：2
作者：
Li, Shaowei [1 ]
Li, Huangyong [1 ]
Cao, Xiufang [1 ]
Chen, Changshui [1 ]
机构：
[1] Huazhong Agr Univ, Coll Sci, Wuhan 430070, Peoples R China
来源：
LETTERS IN DRUG DESIGN & DISCOVERY | 2014年 / 11卷 / 01期
基金：
中国国家自然科学基金;
关键词：
Thiourea; Salicylic acid; Synthesis; Herbicidal activity; Plant growth regulating activity; IN-VITRO; UREA DERIVATIVES; EFFICIENT SYNTHESIS; N-ALKYL; BIOACTIVITY; ANTIBACTERIAL; DESIGN; MOIETY;
D O I：
暂无
中图分类号：
R914 [药物化学];
学科分类号：
100701 ;
摘要：
A series of salicylic acid-oriented thiourea derivatives was conveniently synthesized via multi-steps mainly including alkylation, chlorination, nucleophilic substitution and addition reaction. The structure of all these newly synthesized derivatives was confirmed and characterized by IR, H-1 NMR and MS. The preliminary bioassay indicated that these new compounds have some herbicidal activity or plant growth regulating activity against tested plants.
引用
收藏
页码：98 / 103
页数：6
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