Synthesis and antimicrobial activity of thiazolyl pyrazoles and isoxazoles

被引：29

作者：

Basha, S. S. ^{[1
]}

Divya, K. ^{[1
]}

Padmaja, A. ^{[1
]}

Padmavathi, V. ^{[1
]}

机构：

[1] Sri Venkateswara Univ, Dept Chem, Tirupati 517502, Andhra Pradesh, India

来源：

RESEARCH ON CHEMICAL INTERMEDIATES | 2015年 / 41卷 / 12期

关键词：

Pyrazoles; Isoxazoles; Antibacterial activity; Antifungal activity; BIOLOGICAL EVALUATION; MOIETY; POTENT; INHIBITORS; ANALOGS;

D O I：

10.1007/s11164-015-2013-6

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Thiazolyl pyrazoles and isoxazoles were prepared and their antimicrobial activity studied. Chloro- and nitro-substituted thiazolyl isoxazoles were potential antibacterial agents against Staphylococcus aureus, and nitro-substituted thiazolyl pyrazole was a potential antifungal agent against Aspergillus niger.

引用

页码：10067 / 10083

页数：17

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