International Union of Pharmacology. LXV. The pharmacology and classification of the nuclear receptor superfamily: Glucocorticoid, mineralocorticoid, progesterone, and androgen receptors

被引:320
作者
Lu, Nick Z.
Wardell, Suzanne E.
Burnstein, Kerry L.
Defranco, Donald
Fuller, Peter J.
Giguere, Vincent
Hochberg, Richard B.
McKay, Lorraine
Renoir, Jack-Michel
Weigel, Nancy L.
Wilson, Elizabeth M.
McDonnell, Donald P.
Cidlowski, John A.
机构
[1] NIEHS, Mol Endocrinol Grp, Lab Signal Transduct, NIH,Dept Hlth & Human Serv, Res Triangle Pk, NC 27709 USA
[2] Duke Univ, Med Ctr, Durham, NC USA
[3] Univ Miami, Miller Sch Med, Dept Mol & Cellular Pharmacol, Miami, FL 33152 USA
[4] Univ Pittsburgh, Sch Med, Dept Pharmacol, Pittsburgh, PA 15261 USA
[5] Prince Henrys Inst Med Res, Clayton, Vic, Australia
[6] Royal Victoria Hosp, Mol Oncol Grp, Montreal, PQ H3A 1A1, Canada
[7] Yale Univ, Sch Med, New Haven, CT USA
[8] Bristol Myers Squibb Co, Immune Cell Funct Grp, Princeton, NJ USA
[9] Univ Paris Sud, CNRS, UMR 8612, Chatenay Malabry, France
[10] Baylor Coll Med, Dept Mol & Cellular Biol, Houston, TX 77030 USA
[11] Univ N Carolina, Dept Pediat, Chapel Hill, NC USA
[12] Univ N Carolina, Dept Biochem & Biophys, Chapel Hill, NC USA
关键词
D O I
10.1124/pr.58.4.9
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
[No abstract available]
引用
收藏
页码:782 / 797
页数:16
相关论文
共 109 条
[1]  
Amasheh S, 2000, ANN NY ACAD SCI, V915, P92
[2]   CLONING OF HUMAN MINERALOCORTICOID RECEPTOR COMPLEMENTARY-DNA - STRUCTURAL AND FUNCTIONAL KINSHIP WITH THE GLUCOCORTICOID RECEPTOR [J].
ARRIZA, JL ;
WEINBERGER, C ;
CERELLI, G ;
GLASER, TM ;
HANDELIN, BL ;
HOUSMAN, DE ;
EVANS, RM .
SCIENCE, 1987, 237 (4812) :268-275
[3]   The backdoor pathway to dihydrotestosterone [J].
Auchus, RJ .
TRENDS IN ENDOCRINOLOGY AND METABOLISM, 2004, 15 (09) :432-438
[4]   GLUCOCORTICOID RESISTANCE IN ASTHMA [J].
BARNES, PJ ;
GREENING, AP ;
CROMPTON, GK .
AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 1995, 152 (06) :S125-S140
[5]   DETECTION OF CORTICOSTEROID TYPE-I BINDING-SITES IN HEART [J].
BARNETT, CA ;
PRITCHETT, EL .
MOLECULAR AND CELLULAR ENDOCRINOLOGY, 1988, 56 (03) :191-198
[6]   Mineralocorticoid receptor knockout mice:: Pathophysiology of Na+ metabolism [J].
Berger, S ;
Bleich, M ;
Schmid, W ;
Cole, TJ ;
Peters, J ;
Watanabe, H ;
Kriz, W ;
Warth, R ;
Greger, R ;
Schütz, G .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1998, 95 (16) :9424-9429
[7]  
Bevan CL, 1999, MOL CELL BIOL, V19, P8383
[8]   A ligand-mediated hydrogen bond network required for the activation of the mineralocorticoid receptor [J].
Bledsoe, RK ;
Madauss, KP ;
Holt, JA ;
Apolito, CJ ;
Lambert, MH ;
Pearce, KH ;
Stanley, TB ;
Stewart, EL ;
Trump, RP ;
Willson, TM ;
Williams, SP .
JOURNAL OF BIOLOGICAL CHEMISTRY, 2005, 280 (35) :31283-31293
[9]   Crystal structure of the glucocorticoid receptor ligand binding domain reveals a novel mode of receptor dimerization and coactivator recognition [J].
Bledsoe, RK ;
Montana, VG ;
Stanley, TB ;
Delves, CJ ;
Apolito, CJ ;
McKee, DD ;
Consler, TG ;
Parks, DJ ;
Stewart, EL ;
Willson, TM ;
Lambert, MH ;
Moore, JT ;
Pearce, KH ;
Xu, HE .
CELL, 2002, 110 (01) :93-105
[10]   IDENTIFICATION OF A SPLICE VARIANT OF THE RAT AND HUMAN MINERALOCORTICOID RECEPTOR GENES [J].
BLOEM, LJ ;
GUO, CL ;
PRATT, JH .
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY, 1995, 55 (02) :159-162