Synthesis of Celecoxib, its Pro-drugs and Radiolabeled Derivatives. A Brief Review

被引：5
作者：
Shang, You [1 ]
Du, Jiadi [2 ]
Cui, Hong [3 ]
机构：
[1] Liaoning Med Univ, Affiliated Hosp 1, Dept Anesthesiol, Jinzhou 121001, Liaoning, Peoples R China
[2] Shanghai East Hosp, Dept Obstet & Gynecol, Shanghai 200120, Peoples R China
[3] Peking Univ, Hosp 1, Antiinfect Ward, Inst Clin Pharmacol, Beijing 100034, Peoples R China
来源：
ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL | 2014年 / 46卷 / 02期
关键词：
NITRIC-OXIDE RELEASE; CATALYZED DIRECT ARYLATION; DONOR ESTER PRODRUGS; SELECTIVE COX-2 INHIBITORS; COLORECTAL-CANCER; BIOLOGICAL EVALUATION; NITRATE TOLERANCE; CYCLOOXYGENASE-2; INHIBITOR; EMISSION-TOMOGRAPHY; RAPID METHYLATION;
D O I：
10.1080/00304948.2014.884371
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
[No abstract available]
引用
收藏
页码：132 / 151
页数：20
相关论文
共 83 条
[21]   Proton abstraction mechanism for the palladium-catalyzed intramolecular arylation [J].
García-Cuadrado, D ;
Braga, AAC ;
Maseras, F ;
Echavarren, AM .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2006, 128 (04) :1066-1067
[22]   The Medicinal Chemistry Implications of the Anticancer Effects of Aspirin and Other NSAIDs [J].
Gardiner, P. S. ;
Gilmer, J. F. .
MINI-REVIEWS IN MEDICINAL CHEMISTRY, 2003, 3 (05) :461-470
[23]  
Gately ST, 2005, PROG DRUG RES, V63, P207
[24]   A novel three-step synthesis of Celecoxib via palladium-catalyzed direct arylation [J].
Gaulier, Steven M. ;
McKay, Reuben ;
Swain, Nigel A. .
TETRAHEDRON LETTERS, 2011, 52 (45) :6000-6002
[25]  
Giovannini MG, 2003, INT J IMMUNOPATH PH, V16, P31
[26]   C-H Bonds as Ubiquitous Functionality: A General Approach to Complex Arylated Pyrazoles via Sequential Regioselective C-Arylation and N-Alkylation Enabled by SEM-Group Transposition [J].
Goikhman, Roman ;
Jacques, Teresa L. ;
Sames, Dalibor .
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2009, 131 (08) :3042-3048
[27]   Receptor and enzyme expression for prostanoid metabolism in colorectal cancer related to tumor tissue PGE2 [J].
Gustafsson, Annika ;
Andersson, Marianne ;
Lagerstedt, Kristina ;
Lonnroth, Christina ;
Nordgren, Svante ;
Lundholm, Kent .
INTERNATIONAL JOURNAL OF ONCOLOGY, 2010, 36 (02) :469-478
[28]  
HABER SB, 1989, Patent No. 4820827
[29]   Luminal delivery and dosing considerations of local celecoxib administration to colorectal cancer [J].
Haupt, Sue ;
Zioni, Tamar ;
Gati, Irith ;
Kleinstern, Jackie ;
Rubinstein, Abraham .
EUROPEAN JOURNAL OF PHARMACEUTICAL SCIENCES, 2006, 28 (03) :204-211
[30]   Synthesis of Tri- and Tetrasubstituted Pyrazoles via Ru(II) Catalysis: Intramolecular Aerobic Oxidative C-N Coupling [J].
Hu, Jiantao ;
Chen, Shi ;
Sun, Yonghui ;
Yang, Jing ;
Rao, Yu .
ORGANIC LETTERS, 2012, 14 (19) :5030-5033
123456789