Synthesis of Celecoxib, its Pro-drugs and Radiolabeled Derivatives. A Brief Review

被引：5
作者：
Shang, You [1 ]
Du, Jiadi [2 ]
Cui, Hong [3 ]
机构：
[1] Liaoning Med Univ, Affiliated Hosp 1, Dept Anesthesiol, Jinzhou 121001, Liaoning, Peoples R China
[2] Shanghai East Hosp, Dept Obstet & Gynecol, Shanghai 200120, Peoples R China
[3] Peking Univ, Hosp 1, Antiinfect Ward, Inst Clin Pharmacol, Beijing 100034, Peoples R China
来源：
ORGANIC PREPARATIONS AND PROCEDURES INTERNATIONAL | 2014年 / 46卷 / 02期
关键词：
NITRIC-OXIDE RELEASE; CATALYZED DIRECT ARYLATION; DONOR ESTER PRODRUGS; SELECTIVE COX-2 INHIBITORS; COLORECTAL-CANCER; BIOLOGICAL EVALUATION; NITRATE TOLERANCE; CYCLOOXYGENASE-2; INHIBITOR; EMISSION-TOMOGRAPHY; RAPID METHYLATION;
D O I：
10.1080/00304948.2014.884371
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
[No abstract available]
引用
收藏
页码：132 / 151
页数：20
相关论文
共 83 条
[1]   Diazen-1-ium-1,2-diolated nitric oxide donor ester prodrugs of 5-(4-hydroxymethylphenyl)-1-(4-aminosulfonylphenyl)-3-trifluoromethyl-1H-pyrazole and its methanesulfonyl analog: Synthesis, biological evaluation and nitric oxide release studies [J].
Abdellatif, Khaled R. A. ;
Chowdhury, Morshed Alam ;
Dong, Ying ;
Velazquez, Carlos ;
Das, Dipankar ;
Suresh, Mavanur R. ;
Knaus, Edward E. .
BIOORGANIC & MEDICINAL CHEMISTRY, 2008, 16 (22) :9694-9698
[2]   Diazen-1-ium-1.2-diolated and nitrooxyethyl nitric oxide donor ester prodrugs of anti-inflammatory (E)-2-(aryl)-3-(4-methanesulfonylphenyl)acrylic acids:: Synthesis, cyclooxygenase inhibition, and nitric oxide release studies [J].
Abdellatif, Khaled R. A. ;
Chowdhury, Morshed Alarn ;
Dong, Ying ;
Chen, Qlao-Hong ;
Knaus, Edward E. .
BIOORGANIC & MEDICINAL CHEMISTRY, 2008, 16 (06) :3302-3308
[3]   Novel (E)-2-(aryl)-3-(4-methanesulfonylphenyl)acrylic ester prodrugs possessing a diazen-1-ium-1,2-diolate moiety:: Design, synthesis, cyclooxygenase inhibition, and nitric oxide release studies [J].
Abdellatif, Khaled R. A. ;
Dong, Ying ;
Chen, Qiao-Hong ;
Chowdhury, Morshed Alam ;
Knaus, Edward E. .
BIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (21) :6796-6801
[4]   Diazen-1-ium-1,2-diolated nitric oxide donor ester prodrugs of 5-(4-carboxymethylphenyl)-1-(4-methanesulfonylphenyl)-3-trifluoromethyl-1H-pyrazole and its aminosulfonyl analog: Synthesis, biological evaluation and nitric oxide release studies [J].
Abdellatif, Khaled R. A. ;
Chowdhury, Morshed Alam ;
Dong, Ying ;
Das, Dipankar ;
Yu, Gang ;
Velazquez, Carlos ;
Suresh, Mavanur R. ;
Knaus, Edward E. .
BIOORGANIC & MEDICINAL CHEMISTRY, 2009, 17 (14) :5182-5188
[5]   Transition-Metal-Catalyzed Direct Arylation of (Hetero)Arenes by C-H Bond Cleavage [J].
Ackermann, Lutz ;
Vicente, Ruben ;
Kapdi, Anant R. .
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, 2009, 48 (52) :9792-9826
[6]   Stereospecific fluorination of 1,3,5-tri-O-benzoyl-α-D-ribofuranose-2-sulfonate esters:: preparation of a versatile intermediate for synthesis of 2′-[18F]-fluoro-arabinonucleosides [J].
Alauddin, MM ;
Conti, PS ;
Mathew, T ;
Fissekis, JD ;
Prakash, GKS ;
Watanabe, KA .
JOURNAL OF FLUORINE CHEMISTRY, 2000, 106 (01) :87-91
[7]   Aryl-aryl bond formation by transition-metal-catalyzed direct arylation [J].
Alberico, Dino ;
Scott, Mark E. ;
Lautens, Mark .
CHEMICAL REVIEWS, 2007, 107 (01) :174-238
[8]  
Ambati V. R. R., 2010, [No title captured], Patent No. [WO 2010095024 A2, 2010095024A2]
[9]  
ANDO K, 1999, Patent No. 9964415
[10]  
Battistone MJ, 2010, CLIN MED INSIGHTS-TH, V2, P245
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