Preclinical Evidence That Trametinib Enhances the Response to Tyrosine Kinase Inhibitors in Acute Myeloid Leukemia

被引:1
|
作者
Martinez-Lopez, Joaquin [1 ]
Linares, Maria [2 ]
Morales, Maria Luz [2 ]
Arenas, Alicia [1 ]
Zagorac, Ivana [3 ]
Ayala, Rosa M. [1 ]
Castro, Nerea [4 ]
Rapado, Inmaculada [5 ]
Quintela-Fandino, Miguel [3 ]
机构
[1] Octubre Hosp, Dept Hematol, Madrid, Spain
[2] Hosp 12 Octubre, Inst Invest, Madrid, Spain
[3] Ctr Nacl Invest Oncol, Madrid, Spain
[4] Hosp Octubre, Ser Hematol, Madrid, Spain
[5] Hosp Univ 12 Octubre, Madrid, Spain
关键词
D O I
10.1182/blood.V128.22.1581.1581
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
1581
引用
收藏
页数:4
相关论文
共 50 条
  • [21] New tyrosine kinase inhibitors in chronic myeloid leukemia
    Kantarjian, Hagop
    Cortes, Jorge
    CANCER INVESTIGATION, 2007, 25 : 41 - 43
  • [22] Inhibition of Xanthine Oxidoreductase Enhances the Potential of Tyrosine Kinase Inhibitors against Chronic Myeloid Leukemia
    Romo-Gonzalez, Marta
    Moreno-Paz, Sara
    Garcia-Hernandez, Violeta
    Sanchez-Guijo, Fermin
    Hernandez-Hernandez, Angel
    ANTIOXIDANTS, 2020, 9 (01)
  • [23] Preclinical efficacy for a novel tyrosine kinase inhibitor, ArQule 531 against acute myeloid leukemia
    Elgamal, Ola A.
    Mehmood, Abeera
    Jeon, Jae Yoon
    Carmichael, Bridget
    Lehman, Amy
    Orwick, Shelley J.
    Truxall, Jean
    Goettl, Virginia M.
    Wasmuth, Ronni
    Tran, Minh
    Mitchell, Shaneice
    Lapalombella, Rosa
    Eathiraj, Sudharshan
    Schwartz, Brian
    Stegmaier, Kimberly
    Baker, Sharyn D.
    Hertlein, Erin
    Byrd, John C.
    JOURNAL OF HEMATOLOGY & ONCOLOGY, 2020, 13 (01)
  • [24] Preclinical efficacy for a novel tyrosine kinase inhibitor, ArQule 531 against acute myeloid leukemia
    Ola A. Elgamal
    Abeera Mehmood
    Jae Yoon Jeon
    Bridget Carmichael
    Amy Lehman
    Shelley J. Orwick
    Jean Truxall
    Virginia M. Goettl
    Ronni Wasmuth
    Minh Tran
    Shaneice Mitchell
    Rosa Lapalombella
    Sudharshan Eathiraj
    Brian Schwartz
    Kimberly Stegmaier
    Sharyn D. Baker
    Erin Hertlein
    John C. Byrd
    Journal of Hematology & Oncology, 13
  • [25] Significant preclinical antileukemic activity of the tyrosine kinase inhibitor BVT I in acute myeloid leukemia
    Eriksson, S.
    Hassan, S.
    Hoglund, M.
    Larsson, R.
    Lindhagen, E.
    Aleskog, A.
    Lothgren, A.
    Fohlenhag, K.
    Jensen, A. Jenmalm
    Parrow, V.
    HAEMATOLOGICA-THE HEMATOLOGY JOURNAL, 2007, 92 : 114 - 115
  • [26] Multitargeted tyrosine kinase inhibitors in regulation of growth and survival of acute myeloid leukemia cells
    Lasota, M.
    Balwierz, W.
    FEBS JOURNAL, 2014, 281 : 488 - 488
  • [27] Gold nanoparticles enhance the effect of tyrosine kinase inhibitors in acute myeloid leukemia therapy
    Petrushev, Bobe
    Boca, Sanda
    Simon, Timea
    Berce, Cristian
    Frinc, Ioana
    Dima, Delia
    Selicean, Sonia
    Gafencu, Grigore-Aristide
    Tanase, Alina
    Zdrenghea, Mihnea
    Florea, Adrian
    Suarasan, Sorina
    Dima, Liana
    Stanciu, Raluca
    Jurj, Ancuta
    Buzoianu, Anca
    Cucuianu, Andrei
    Astilean, Simion
    Irimie, Alexandru
    Tomuleasa, Ciprian
    Berindan-Neagoe, Ioana
    INTERNATIONAL JOURNAL OF NANOMEDICINE, 2016, 11 : 641 - 660
  • [28] Antitumor efficacy of arsenic/interferon in preclinical models of chronic myeloid leukemia resistant to tyrosine kinase inhibitors
    El Eit, Rabab
    Itani, Abdul Rahman
    Nassar, Farah
    Rasbieh, Nagham
    Jabbour, Mark
    Santina, Ahmad
    Zaatari, Ghazi
    Mahon, Francois-Xavier
    Bazarbachi, Ali
    Nasr, Rihab
    CANCER, 2019, 125 (16) : 2818 - 2828
  • [29] Microenvironmental Factors Determine the Sensitivity of Acute Myeloid Leukemia Cells to Tyrosine Kinase Inhibitors
    Shimada, Akira
    Orwick, Shelley
    Fujisaki, Hiroyuki
    Campana, Dario
    Baker, Sharyn D.
    BLOOD, 2008, 112 (11) : 576 - 576
  • [30] FMS-Like Tyrosine Kinase 3 Inhibitors for the Treatment of Acute Myeloid Leukemia
    Novatcheva, Elli D.
    Anouty, Yasmine
    Saunders, Ila
    Mangan, James K.
    Goodman, Aaron M.
    CLINICAL LYMPHOMA MYELOMA & LEUKEMIA, 2022, 22 (03): : E161 - E184