A New Method for the Synthesis of 3-Substituted Indoles

被引：14
作者：
Natarajan, Rakesh [1 ]
Rappai, John P. [2 ]
Unnikrishnan, Peruparampil A. [1 ]
Radhamani, Sandhya [3 ]
Prathapan, Sreedharan [1 ]
机构：
[1] Cochin Univ Sci & Technol, Dept Appl Chem, Kochi 682022, Kerala, India
[2] Govt Victoria Coll, Dept Chem, Palakkad 678001, India
[3] NSS Coll, Dept Chem, Ottapalam 679103, Palakkad, India
来源：
SYNLETT | 2015年 / 26卷 / 17期
关键词：
indoles; nitrones; electron-deficient acetylenes; nucleophilic addition; 1,3-dipolar additions; NONREARRANGED MONOTERPENOID UNIT; PALLADIUM-CATALYZED REACTIONS; SOLID-PHASE SYNTHESIS; 2,3-DISUBSTITUTED INDOLES; C3-QUATERNARY INDOLENINES; ISOCYANIDE INSERTION; BIOLOGICAL-ACTIVITY; DERIVATIVES; NITRONES; ALKALOIDS;
D O I：
10.1055/s-0035-1560210
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Starting from readily accessible nitrones and electron-deficient acetylenes, a highly efficient and versatile synthetic protocol for 3-substituted indoles has been developed.
引用
收藏
页码：2467 / 2471
页数：5
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