4-Thiazolidinones: The advances continue ...

被引:283
作者
Tripathi, Avinash C. [1 ]
Gupta, Shiv Ji [1 ]
Fatima, Gul Naz [1 ]
Sonar, Pankaj Kumar [1 ]
Verma, Amit [2 ]
Saraf, Shailendra K. [1 ]
机构
[1] Babu Banarasi Das Northern India Inst Technol, Fac Pharm, Dept Pharmaceut Chem, Lucknow 226028, Uttar Pradesh, India
[2] Maharaja Sayajirao Univ Baroda, Fac Engn & Technol, Dept Pharm, Vadodara 390001, Gujarat, India
关键词
Thiazolidin-4-ones; Synthesis and characterization; Stereochemistry; Anticancer; Antiviral; Anticonvulsant; Cardiovascular; NSAID; Antidiabetic; Antihyperlipidemic; Antimicrobial; Antituberculosis; Antiparasitic; Patents on 4-thiazolidinones; FOLLICLE-STIMULATING-HORMONE; MICROWAVE-ASSISTED SYNTHESIS; CALCIUM OVERLOAD INHIBITION; ONE-POT SYNTHESIS; BIOLOGICAL EVALUATION; ANTIMICROBIAL ACTIVITY; ANTICONVULSANT ACTIVITY; ANTI-HIV; THIAZOLIDINONE DERIVATIVES; ANTITUMOR-ACTIVITY;
D O I
10.1016/j.ejmech.2013.11.017
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
The diversity in the biological response of 4-thiazolidinones has attracted the attention of many researchers to explore this framework for its potential. It is, therefore, of prime importance that the study of this topic and the development of new synthetic strategies should be based on the most recent knowledge, emerging from the latest research. This review is an endeavor to highlight the progress in the chemistry and biological activity of the 4-thiazolidinones, predominantly after 2006. The last section of the review encompasses the various patents granted on 4-thiazolidinone analogs/derivatives with World Intellectual Proprietary Organization (WIPO) and United State Patent Trademark Office (USPTO), particularly in the duration of the year 2000 to the year 2012. (C) 2013 Elsevier Masson SAS. All rights reserved.
引用
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页码:52 / 77
页数:26
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