Regiospecific functionalization of indole-2-carboxylates and diastereoselective preparation of the corresponding indolines

被引：0
|
作者：
Collot, V [1 ]
Schmitt, M [1 ]
Marwah, P [1 ]
Bourguignon, JJ [1 ]
机构：
[1] Fac Pharm, Lab Pharmacochim Commun Cellulaire, ERS 655, F-67401 Illkirch Graffenstaden, France
来源：
HETEROCYCLES | 1999年 / 51卷 / 12期
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The N-acyl derivatives of 3-substituted indole-2-carboxylates prepared through several routes were submitted to catalytic hydrogenation affording either cis- or trans-indoline diastereomers after quantitative C-2 epimerization.
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页码：2823 / 2847
页数：25
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