3-[2-(pyrrolidin-1-yl)ethyl]indoles and 3-[3-(piperidin-1-yl)propyl]indoles: Agonists for the h5-HT1D receptor with high selectivity over the h5-HT1B subtype

被引:17
作者
Castro, JL [1 ]
Street, LJ [1 ]
Guiblin, AR [1 ]
Jelley, RA [1 ]
Russell, MGN [1 ]
Sternfeld, F [1 ]
Beer, MS [1 ]
Stanton, JA [1 ]
Matassa, VG [1 ]
机构
[1] MERCK SHARP & DOHME LTD,RES LABS,NEUROSCI RES CTR,DEPT BIOCHEM,HARLOW CM20 2QR,ESSEX,ENGLAND
关键词
D O I
10.1021/jm9704558
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:3497 / 3500
页数:6
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