ZrCl4-mediated synthesis of 1,2,3-triazoles from vinyl nitrates and their biological evaluation

被引：3
作者：
Sridhar, Gattu [1 ]
Somnath, Mudavath [1 ]
Sharma, Gangavaram V. M. [1 ]
Prashanth, Thodupunuri [1 ]
机构：
[1] Indian Inst Chem Technol, CSIR, Organ & Biomol Chem Div, Hyderabad 500107, Andhra Pradesh, India
来源：
SYNTHETIC COMMUNICATIONS | 2017年 / 47卷 / 06期
关键词：
1,2,3-Triazoles; CH3NO2; vinyl nitrates; zirconium(IV)chloride; 1,3-DIPOLAR CYCLOADDITION; RATIONAL DESIGN; RECENT TRENDS; INHIBITORS; CHEMISTRY; AZIDES; ZRCL4;
D O I：
10.1080/00397911.2016.1270324
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
A ZrCl4-mediated simple method for the conversion of vinyl nitrates to 1,2,3-triazoles in excellent yields is developed. The obtained new triazoles were evaluated for their antimicrobial activity.
引用
收藏
页码：551 / 556
页数：6
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