Efficient and regiospecific one-pot synthesis of substituted 1,2,4-triazoles

被引：80

作者：

Stocks, MJ ^{[1
]}

Cheshire, DR ^{[1
]}

Reynolds, R ^{[1
]}

机构：

[1] AstraZeneca R&D Charnwood, Dept Med Chem, Loughborough LE11 5RH, Leics, England

来源：

ORGANIC LETTERS | 2004年 / 6卷 / 17期

关键词：

D O I：

10.1021/ol048863a

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

An efficient one-pot, three-component synthesis of substituted 1,2,4-triazoles has been developed, utilizing a wide range of substituted primary amines and acyl hydrazides.

引用

页码：2969 / 2971

页数：3

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