Chiral histone deacetylase inhibitors: Synthesis and biological evaluation

被引：0
|
作者：
Onate, Alma [1 ]
Tucker, Janelle [1 ]
Hogle, Emily [1 ]
Do, Thuy [1 ]
Thowfeik, Fathima [2 ]
Merino, Edward [2 ]
Ma, Lili [1 ]
机构：
[1] Northern Kentucky Univ, Chem, Hamilton, OH USA
[2] Univ Cincinnati, Chem, Cincinnati, OH USA
来源：
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2016年 / 251卷
关键词：
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
1144
引用
收藏
页数：1
相关论文
共 50 条
  • [31] Design, Synthesis, and Biological Activity of Hydroxamic Tertiary Amines as Histone Deacetylase Inhibitors
    Terracciano, Stefania
    Chini, Maria Giovanna
    Riccio, Raffaele
    Bruno, Ines
    Bifulco, Giuseppe
    CHEMMEDCHEM, 2012, 7 (04) : 694 - 702
  • [32] Synthesis and Biological Studies of New Histone Deacetylase Inhibitors Containing the Dihydroquinazolinone Cycle
    Kolotaev, A., V
    Osipov, V. N.
    Balaev, A. N.
    Okhmanovich, K. A.
    Vartanyan, A. A.
    Khochenkov, D. A.
    Matevosyan, K. R.
    Khochenkova, U. A.
    Khachatryan, D. S.
    MODERN SYNTHETIC METHODOLOGIES FOR CREATING DRUGS AND FUNCTIONAL MATERIALS (MOSM2019), 2020, 2280
  • [33] Synthesis and biological properties of novel, uracil-containing histone deacetylase inhibitors
    Mai, Antonello
    Massa, Silvio
    Rotili, Dante
    Simeoni, Silvia
    Ragno, Rino
    Botta, Giorgia
    Nebbioso, Angela
    Miceli, Marco
    Altucci, Lucia
    Brosch, Gerald
    JOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (20) : 6046 - 6056
  • [34] MEDI 148-Synthesis and evaluation of cyclopeptide inhibitors of histone deacetylase
    Marson, Charles M.
    Sengmany, Stephane
    Middleton, Brian
    Dines, Jonathan
    Thomas, N. Shaun B.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2006, 232
  • [35] Synthesis and pharmacological evaluation of histone deacetylase inhibitors as fetal hemoglobin inducers
    Dos Santos, Jean
    Melchior, Aylime
    Bosquesi, Priscila
    Pavan, Aline
    Lanaro, Carolina
    Chung, ManChin
    Rusinova, Radda
    Chelucci, Rafael
    Andersen, Olaf
    Costa, Fernando
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 255
  • [36] Design, Synthesis, Biological Evaluation, and Structural Characterization of Potent Histone Deacetylase Inhibitors Based on Cyclic α/β-Tetrapeptide Architectures
    Montero, Ana
    Beierle, John M.
    Olsen, Christian A.
    Ghadiri, M. Reza
    JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, 2009, 131 (08) : 3033 - 3041
  • [37] Synthesis and biological evaluation of selective histone deacetylase 6 inhibitors as multifunctional agents against Alzheimer's disease
    Wang, Xiu-Xiu
    Xie, Fei
    Jia, Cong-Cong
    Yan, Ning
    Zeng, Yan-Li
    Wu, Jing-De
    Liu, Zhao-Peng
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 225
  • [38] Synthesis and Biological Evaluation of Novel Thiazolyl-Coumarin Derivatives as Potent Histone Deacetylase Inhibitors with Antifibrotic Activity
    Pardo-Jimenez, Viviana
    Navarrete-Encina, Patricio
    Diaz-Araya, Guillermo
    MOLECULES, 2019, 24 (04):
  • [39] Design, Synthesis and Biological Evaluation of Nitro Oxide Donating N-Hydroxycinnamamide Derivatives as Histone Deacetylase Inhibitors
    Tu, Shiliang
    Yuan, Hang
    Hu, Jie
    Zhao, Chengguang
    Chai, Rui
    Cao, Hongfeng
    CHEMICAL & PHARMACEUTICAL BULLETIN, 2014, 62 (12) : 1185 - 1191
  • [40] Oxime Amides as a Novel Zinc Binding Group in Histone Deacetylase Inhibitors: Synthesis, Biological Activity, and Computational Evaluation
    Botta, Cinzia B.
    Cabri, Walter
    Cini, Elena
    De Cesare, Lucia
    Fattorusso, Caterina
    Giannini, Giuseppe
    Persico, Marco
    Petrella, Antonello
    Rondinelli, Francesca
    Rodriquez, Manuela
    Russo, Adele
    Taddei, Maurizio
    JOURNAL OF MEDICINAL CHEMISTRY, 2011, 54 (07) : 2165 - 2182
12345