Quaternary ammonium salt as alkylation agent in three-component reactions for the synthesis of benzothiazoles in water

被引：8
|
作者：
Pan, Lei [1 ]
Yu, Lintao [1 ,2 ]
Wu, Zhiqing [1 ]
Li, Zhengkai [1 ]
Xiang, Haifeng [1 ]
Zhou, Xiangge [1 ]
机构：
[1] Sichuan Univ, Coll Chem, Inst Homogeneous Catalysis, Chengdu 610064, Peoples R China
[2] Nanyang Normal Univ, Coll Chem & Pharmaceut Engn, Nanyang 473061, Peoples R China
来源：
RSC ADVANCES | 2014年 / 4卷 / 53期
关键词：
STREPTOMYCES SP 517-02; SUBSTITUTED BENZOTHIAZOLES; 2-SUBSTITUTED BENZOTHIAZOLES; INTRAMOLECULAR CYCLIZATION; ANTITUMOR BENZOTHIAZOLES; MULTICOMPONENT REACTIONS; CYTOTOXIC METABOLITE; PARALLEL SYNTHESIS; BENZOXAZOLES; COPPER;
D O I：
10.1039/c4ra04145c
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Substituted benzothiazoles are synthesized by metal-catalyst-free three-component reactions of o-iodoaniline, quaternary ammonium salt, and sulfur powder in water with moderate-to-excellent yields up to 95%.
引用
收藏
页码：27775 / 27779
页数：5
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