Closing the Loop: Developing an Integrated Design, Make, and Test Platform for Discovery

被引:21
作者
Parry, David M. [1 ]
机构
[1] Cyclofluidic Ltd, BioPark, Broadwater Rd, Welwyn Garden City AL7 3AX, Herts, England
来源
ACS MEDICINAL CHEMISTRY LETTERS | 2019年 / 10卷 / 06期
基金
“创新英国”项目;
关键词
Automated Discovery; Design Make and Test; Integration; Flow Synthesis; ABL1; Kinase; INHIBITORS; OPTIMIZATION; DIVERSE;
D O I
10.1021/acsmedchemlett.9b00095
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
The relatively slow cycle time within medicinal chemistry from synthesis to assay is constantly being challenged to help improve the efficiency of the discovery process. While both synthesis and assay have been automated to varying degrees, there has, until recently, been limited focus on the complete design, make, and test process. This Innovations article outlines the development of Cyclofluidic from inception through to the commercialization of a fully integrated closed loop design, synthesis, and screen platform.
引用
收藏
页码:848 / 856
页数:17
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