Expedient method for the solid-phase synthesis of some 4-substituted-4,5-dihydropyridazin-3(2H)-ones

被引：13

作者：

Gouault, N ^{[1
]}

Cupif, JF ^{[1
]}

Amoros, M ^{[1
]}

David, M ^{[1
]}

机构：

[1] Fac Pharm, UPRES Synthese & Exract Mol Visee Therapeut, F-35043 Rennes, France

来源：

JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1 | 2002年 / 20期

关键词：

D O I：

10.1039/b205607k

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The solid-phase synthesis of some 4-amino- 4,5-dihydropyridazin-3( 2H)-ones has been realised using regiospecific Michael addition and subsequent cyclorelease reactions.

引用

页码：2234 / 2236

页数：3

共 17 条

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