Synthesis, characterization, and antimicrobial activity of new benzofuran derivatives

被引：7

作者：

Kenchappa, R. ^{[1
]}

Bodke, Yadav D. ^{[1
]}

Telkar, Sandeep ^{[2
]}

Sindhe, M. Aruna ^{[1
]}

Giridhar, M. ^{[1
]}

机构：

[1] Kuvempu Univ Shankaraghatta, Dept PG Studies & Res Ind Chem, Shivamogga 577451, Karnataka, India

[2] Kuvempu Univ, Dept PG Studies & Res Biotechnol & Bioinformat, Shankaraghatta 577451, Karnataka, India

来源：

RUSSIAN JOURNAL OF GENERAL CHEMISTRY | 2016年 / 86卷 / 12期

关键词：

benzofuran; meldrums acid; Knoevenagel condensation; antimicrobial; molecular docking; FUSARIUM-EQUISETI; INHIBITORS; ACID;

D O I：

10.1134/S107036321612046X

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

A novel series of (5-substituted-1-benzofuran-2-yl)(2,4-substituted phenyl)methanones (4a-4i) have been prepared by the Knoevenagel condensation of (5-substituted-1-benzofuran-2-yl)(2,4-substituted phenyl)methanone (3a-3i) with Meldrum's acid. The structures of the synthesized compounds were characterized by different spectroscopic techniques. All newly synthesized compounds were screened for antimicrobial activity.

引用

收藏

页码：2827 / 2836

页数：10

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