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NOE pumping. 2. A high-throughput method to determine compounds with binding affinity to macromolecules by NMR
被引:106
作者
:
Chen, AD
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst Biomed Res, Summit, NJ 07901 USA
Novartis Inst Biomed Res, Summit, NJ 07901 USA
Chen, AD
[
1
]
Shapiro, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Novartis Inst Biomed Res, Summit, NJ 07901 USA
Novartis Inst Biomed Res, Summit, NJ 07901 USA
Shapiro, MJ
[
1
]
机构
:
[1]
Novartis Inst Biomed Res, Summit, NJ 07901 USA
来源
:
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY
|
2000年
/ 122卷
/ 02期
关键词
:
D O I
:
10.1021/ja992588j
中图分类号
:
O6 [化学];
学科分类号
:
0703 ;
摘要
:
[No abstract available]
引用
收藏
页码:414 / 415
页数:2
相关论文
共 18 条
[1]
AKI H, 1992, CHEM PHARM BULL, V40, P1553
[2]
A HIGH-TEMPERATURE SUPERCONDUCTING RECEIVER FOR NUCLEAR-MAGNETIC-RESONANCE MICROSCOPY
BLACK, RD
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
BLACK, RD
EARLY, TA
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
EARLY, TA
ROEMER, PB
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
ROEMER, PB
MUELLER, OM
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
MUELLER, OM
MOGROCAMPERO, A
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
MOGROCAMPERO, A
TURNER, LG
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
TURNER, LG
JOHNSON, GA
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
JOHNSON, GA
[J].
SCIENCE,
1993,
259
(5096)
: 793
-
795
[3]
EFFECTS OF DIFFUSION ON FREE PRECESSION IN NUCLEAR MAGNETIC RESONANCE EXPERIMENTS
CARR, HY
论文数:
0
引用数:
0
h-index:
0
CARR, HY
PURCELL, EM
论文数:
0
引用数:
0
h-index:
0
PURCELL, EM
[J].
PHYSICAL REVIEW,
1954,
94
(03):
: 630
-
638
[4]
NOE pumping: A novel NMR technique for identification of compounds with binding affinity to macromolecules
Chen, A
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Chen, A
Shapiro, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Shapiro, MJ
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1998,
120
(39)
: 10258
-
10259
[5]
THEORY OF THE TIME-DEPENDENT TRANSFERRED NUCLEAR OVERHAUSER EFFECT - APPLICATIONS TO STRUCTURAL-ANALYSIS OF LIGAND PROTEIN COMPLEXES IN SOLUTION
CLORE, GM
论文数:
0
引用数:
0
h-index:
0
CLORE, GM
GRONENBORN, AM
论文数:
0
引用数:
0
h-index:
0
GRONENBORN, AM
[J].
JOURNAL OF MAGNETIC RESONANCE,
1983,
53
(03)
: 423
-
442
[6]
THEORY AND APPLICATIONS OF THE TRANSFERRED NUCLEAR OVERHAUSER EFFECT TO THE STUDY OF THE CONFORMATIONS OF SMALL LIGANDS BOUND TO PROTEINS
CLORE, GM
论文数:
0
引用数:
0
h-index:
0
CLORE, GM
GRONENBORN, AM
论文数:
0
引用数:
0
h-index:
0
GRONENBORN, AM
[J].
JOURNAL OF MAGNETIC RESONANCE,
1982,
48
(03)
: 402
-
417
[7]
One-dimensional relaxation- and diffusion-edited NMR methods for screening compounds that bind to macromolecules
Hajduk, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Hajduk, PJ
Olejniczak, ET
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Olejniczak, ET
Fesik, SW
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Fesik, SW
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1997,
119
(50)
: 12257
-
12261
[8]
High-throughput nuclear magnetic resonance-based screening
Hajduk, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Hajduk, PJ
Gerfin, T
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Gerfin, T
Boehlen, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Boehlen, JM
Häberli, M
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Häberli, M
Marek, D
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Marek, D
Fesik, SW
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Fesik, SW
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1999,
42
(13)
: 2315
-
2317
[9]
Detecting binding affinity to immobilized receptor proteins in compound libraries by HR-MAS STD NMR
Klein, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Klein, J
Meinecke, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Meinecke, R
Mayer, M
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Mayer, M
Meyer, B
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Meyer, B
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1999,
121
(22)
: 5336
-
5337
[10]
Diffusion-edited NMR-affinity NMR for direct observation of molecular interactions
Lin, MF
论文数:
0
引用数:
0
h-index:
0
机构:
SANDOZ PHARMACEUT CORP,RES INST,PRECLIN RES,DEPT CENT TECHNOL,E HANOVER,NJ 07936
Lin, MF
Shapiro, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
SANDOZ PHARMACEUT CORP,RES INST,PRECLIN RES,DEPT CENT TECHNOL,E HANOVER,NJ 07936
Shapiro, MJ
Wareing, JR
论文数:
0
引用数:
0
h-index:
0
机构:
SANDOZ PHARMACEUT CORP,RES INST,PRECLIN RES,DEPT CENT TECHNOL,E HANOVER,NJ 07936
Wareing, JR
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1997,
119
(22)
: 5249
-
5250
←
1
2
→
共 18 条
[1]
AKI H, 1992, CHEM PHARM BULL, V40, P1553
[2]
A HIGH-TEMPERATURE SUPERCONDUCTING RECEIVER FOR NUCLEAR-MAGNETIC-RESONANCE MICROSCOPY
BLACK, RD
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
BLACK, RD
EARLY, TA
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
EARLY, TA
ROEMER, PB
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
ROEMER, PB
MUELLER, OM
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
MUELLER, OM
MOGROCAMPERO, A
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
MOGROCAMPERO, A
TURNER, LG
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
TURNER, LG
JOHNSON, GA
论文数:
0
引用数:
0
h-index:
0
机构:
DUKE UNIV,DEPT RADIOL,DURHAM,NC 27710
JOHNSON, GA
[J].
SCIENCE,
1993,
259
(5096)
: 793
-
795
[3]
EFFECTS OF DIFFUSION ON FREE PRECESSION IN NUCLEAR MAGNETIC RESONANCE EXPERIMENTS
CARR, HY
论文数:
0
引用数:
0
h-index:
0
CARR, HY
PURCELL, EM
论文数:
0
引用数:
0
h-index:
0
PURCELL, EM
[J].
PHYSICAL REVIEW,
1954,
94
(03):
: 630
-
638
[4]
NOE pumping: A novel NMR technique for identification of compounds with binding affinity to macromolecules
Chen, A
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Chen, A
Shapiro, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Nova Pharmaceut Corp, Preclin Res, Dept Analyt, Summit, NJ 07901 USA
Shapiro, MJ
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1998,
120
(39)
: 10258
-
10259
[5]
THEORY OF THE TIME-DEPENDENT TRANSFERRED NUCLEAR OVERHAUSER EFFECT - APPLICATIONS TO STRUCTURAL-ANALYSIS OF LIGAND PROTEIN COMPLEXES IN SOLUTION
CLORE, GM
论文数:
0
引用数:
0
h-index:
0
CLORE, GM
GRONENBORN, AM
论文数:
0
引用数:
0
h-index:
0
GRONENBORN, AM
[J].
JOURNAL OF MAGNETIC RESONANCE,
1983,
53
(03)
: 423
-
442
[6]
THEORY AND APPLICATIONS OF THE TRANSFERRED NUCLEAR OVERHAUSER EFFECT TO THE STUDY OF THE CONFORMATIONS OF SMALL LIGANDS BOUND TO PROTEINS
CLORE, GM
论文数:
0
引用数:
0
h-index:
0
CLORE, GM
GRONENBORN, AM
论文数:
0
引用数:
0
h-index:
0
GRONENBORN, AM
[J].
JOURNAL OF MAGNETIC RESONANCE,
1982,
48
(03)
: 402
-
417
[7]
One-dimensional relaxation- and diffusion-edited NMR methods for screening compounds that bind to macromolecules
Hajduk, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Hajduk, PJ
Olejniczak, ET
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Olejniczak, ET
Fesik, SW
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Fesik, SW
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1997,
119
(50)
: 12257
-
12261
[8]
High-throughput nuclear magnetic resonance-based screening
Hajduk, PJ
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Hajduk, PJ
Gerfin, T
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Gerfin, T
Boehlen, JM
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Boehlen, JM
Häberli, M
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Häberli, M
Marek, D
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Marek, D
Fesik, SW
论文数:
0
引用数:
0
h-index:
0
机构:
Abbott Labs, Div Pharmaceut Discovery, Abbott Pk, IL 60064 USA
Fesik, SW
[J].
JOURNAL OF MEDICINAL CHEMISTRY,
1999,
42
(13)
: 2315
-
2317
[9]
Detecting binding affinity to immobilized receptor proteins in compound libraries by HR-MAS STD NMR
Klein, J
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Klein, J
Meinecke, R
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Meinecke, R
Mayer, M
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Mayer, M
Meyer, B
论文数:
0
引用数:
0
h-index:
0
机构:
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Univ Hamburg, Inst Organ Chem, D-20146 Hamburg, Germany
Meyer, B
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1999,
121
(22)
: 5336
-
5337
[10]
Diffusion-edited NMR-affinity NMR for direct observation of molecular interactions
Lin, MF
论文数:
0
引用数:
0
h-index:
0
机构:
SANDOZ PHARMACEUT CORP,RES INST,PRECLIN RES,DEPT CENT TECHNOL,E HANOVER,NJ 07936
Lin, MF
Shapiro, MJ
论文数:
0
引用数:
0
h-index:
0
机构:
SANDOZ PHARMACEUT CORP,RES INST,PRECLIN RES,DEPT CENT TECHNOL,E HANOVER,NJ 07936
Shapiro, MJ
Wareing, JR
论文数:
0
引用数:
0
h-index:
0
机构:
SANDOZ PHARMACEUT CORP,RES INST,PRECLIN RES,DEPT CENT TECHNOL,E HANOVER,NJ 07936
Wareing, JR
[J].
JOURNAL OF THE AMERICAN CHEMICAL SOCIETY,
1997,
119
(22)
: 5249
-
5250
←
1
2
→