SUPPRESSION OF CYTOCHROME P450 3A4 ACTIVITY BY UDP-GLUCURONOSYLTRANSFERASE (UGT) 2B7: THE ROLE OF CHARGED RESIDUE(S) IN THE CYTOSOLIC TAIL OF UGT2B7

被引:0
作者
Miyauchi, Yuu [1 ]
Ishii, Yuji [1 ]
Nagata, Kiyoshi [2 ]
Yamazoe, Yasushi [3 ]
Mackenzie, Peter I. [4 ,5 ]
Yamada, Hideyuki [1 ]
机构
[1] Kyushu Univ, Grad Sch Pharmaceut Sci, Lab Mol Life Sci, Fukuoka 812, Japan
[2] Tohoku Pharmaceut Univ, Sendai, Miyagi, Japan
[3] Govt Japan, Cabinet Off, Food Safety Commiss, Tokyo, Japan
[4] Flinders Med Ctr, Dept Clin Pharmacol, Adelaide, SA, Australia
[5] Flinders Univ S Australia, Adelaide, SA 5001, Australia
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D O I
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中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
A1
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页码:34 / 34
页数:1
相关论文
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[1]   Interaction of Cytochrome P450 3A4 and UDP-Glucuronosyltransferase 2B7: Evidence for Protein-Protein Association and Possible Involvement of CYP3A4 J-Helix in the Interaction [J].
Takeda, Shuso ;
Ishii, Yuji ;
Iwanaga, Megumi ;
Nurrochmad, Arief ;
Ito, Yuji ;
Mackenzie, Peter I. ;
Nagata, Kiyoshi ;
Yamazoe, Yasushi ;
Oguri, Kazuta ;
Yamada, Hideyuki .
MOLECULAR PHARMACOLOGY, 2009, 75 (04) :956-964