Case History: Chantix™/Champix™ (Varenicline Tartrate), a Nicotinic Acetylcholine Receptor Partial Agonist as a Smoking Cessation Aid

被引:21
作者
Coe, Jotham W. [1 ]
Rollema, Hans [1 ]
O'Neill, Brian T. [1 ]
机构
[1] Pfizer Global Res & Dev, Groton Labs, Groton, CT 06340 USA
来源
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 44 | 2009年 / 44卷
关键词
RANDOMIZED CONTROLLED-TRIAL; 10-SUBSTITUTED CYTISINE DERIVATIVES; SUSTAINED-RELEASE BUPROPION; DISCRIMINATIVE STIMULUS; DOSE PHARMACOKINETICS; CHOLINERGIC-RECEPTOR; HEALTHY SMOKERS; BETA-2; SUBUNIT; IN-VIVO; (-)-CYTISINE;
D O I
10.1016/S0065-7743(09)04404-2
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:71 / +
页数:32
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