An Updated Coverage on the Synthesis of Benzo[b]thiophenes via Transition-metal-catalyzed Reactions: A Review

被引：7

作者：

Ejaz, Saba ^{[1
]}

Zubair, Muhammad ^{[1
]}

Rizwan, Komal ^{[1
,2
]}

Karakaya, Idris ^{[3
]}

Rasheed, Tahir ^{[4
]}

Rasool, Nasir ^{[1
]}

机构：

[1] Govt Coll Univ, Dept Chem, Faisalabad 38000, Pakistan

[2] Univ Sahiwal, Dept Chem, Sahiwal 57000, Pakistan

[3] Gebze Tech Univ, Coll Basic Sci, Dept Chem, TR-41400 Gebze, Turkey

[4] Shanghai Jiao Tong Univ, Sch Chem & Chem Engn, Shanghai 200240, Peoples R China

来源：

CURRENT ORGANIC CHEMISTRY | 2021年 / 25卷 / 01期

关键词：

Benno[b]thiophene; couplings; transition metals; heterocyclics; palladium; synthesis; ONE-POT SYNTHESIS; HETERO-FUSED ANALOGS; SUBSEQUENT 6-PI-ELECTROCYCLIZATION REACTIONS; C-H ACTIVATION; BOND FORMATION; FUNCTIONALIZED BENZOTHIOPHENES; ELECTROPHILIC CYCLIZATION; EFFICIENT SYNTHESIS; 2,3-DISUBSTITUTED BENZOTHIOPHENES; INTERMOLECULAR CYCLIZATION;

D O I：

10.2174/1385272824999201111204317

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The benzo[b]thiophene nucleus is ubiquitous in biologically and pharmaceutically important compounds. These moieties are highly important in materials science. The synthesis of benzothiophene as a privileged structure has readily become a subject of great interest and actively pursued in recent years. This review focuses on facile and convenient methods of synthesis of benzo[b]thiophene based molecules through different transition metals catalyzed reactions.

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页码：40 / 67

页数：28

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