Discovery and evaluation of selective, orally available and brain penetrant inhibitors of leucine rich repeat kinase 2 (LRRK2)

被引:0
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作者
DeMong, Duane [1 ]
Basu, Kallol [1 ]
Scott, Jack [1 ]
Miller, Michael [1 ]
Agnihotri, Gautam [1 ]
Baptista, Marco [1 ]
Cheewatrakoolpong, Boonlert [1 ]
Columbus, John [1 ]
Dai, Xing [1 ]
Duan, Xiaobang [2 ]
Fell, Matthew [1 ]
Frank, Emily [1 ]
Frassetto, Andrea [1 ]
Greshock, Thomas [1 ]
Harris, Joel [1 ]
Hruza, Alan [1 ]
Hu, Zhiyong [1 ]
Li, Wei [1 ]
Lin, Sue-Ing [1 ]
Liu, Hong [1 ]
Macala, Megan [1 ]
Mei, Hong [1 ]
Mirescu, Christian [1 ]
Morrow, John [1 ]
Poirier, Marc [1 ]
Scapin, Giovanna [1 ]
Sherborne, Bradley [1 ]
Smith, Michelle [1 ]
Stevenson, Heather [1 ]
Strickland, Corey [1 ]
Tempest, Paul [2 ]
Vicarel, Monica [1 ]
Walsh, Paul [1 ]
Xiao, Li [1 ]
Zhang, Honglu [1 ]
Zhou, Xiaoping [1 ]
Duffy, Joseph [1 ]
Kennedy, Matthew [1 ]
McCauley, John [1 ]
Nargund, Ravi [1 ]
Parker, Eric [1 ]
Ruck, Rebecca [1 ]
Stamford, Andrew [1 ]
Weber, Ann [1 ]
机构
[1] Merck & Co Inc, Merck Res Labs, Somerset, NJ USA
[2] Shanghai Chempartner, Shanghai, Peoples R China
关键词
D O I
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中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
19
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页数:1
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