Agonist binding to G-protein coupled receptors

被引:5
作者
Strange, PG [1 ]
机构
[1] Univ Reading, Sch Anim & Microbial Sci, Reading RG6 6AJ, Berks, England
关键词
G-protein coupled receptors; agonist binding; receptor theory; receptor activation;
D O I
10.1038/sj.bjp.0702991
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
引用
收藏
页码:820 / 821
页数:2
相关论文
共 17 条
[1]   Functional microdomains in g-protein-coupled receptors - The conserved Arginine-cage motif in the gonadotropin-releasing hormone receptor [J].
Ballesteros, J ;
Kitanovic, S ;
Guarnieri, F ;
Davies, P ;
Fromme, BJ ;
Konvicka, K ;
Chi, L ;
Millar, RP ;
Davidson, JS ;
Weinstein, H ;
Sealfon, SC .
JOURNAL OF BIOLOGICAL CHEMISTRY, 1998, 273 (17) :10445-10453
[2]  
CHUNG FZ, 1988, J BIOL CHEM, V263, P4052
[3]  
Colquhoun D, 1998, BRIT J PHARMACOL, V125, P924
[4]  
FRASER CM, 1989, MOL PHARMACOL, V36, P840
[5]  
HORSTMAN DA, 1990, J BIOL CHEM, V265, P21590
[6]   CONSTITUTIVE ACTIVITY OF RECEPTORS COUPLED TO GUANINE-NUCLEOTIDE REGULATORY PROTEINS [J].
LEFKOWITZ, RJ ;
COTECCHIA, S ;
SAMAMA, P ;
COSTA, T .
TRENDS IN PHARMACOLOGICAL SCIENCES, 1993, 14 (08) :303-307
[7]  
NEVE KA, 1991, MOL PHARMACOL, V39, P733
[8]  
SAMAMA P, 1993, J BIOL CHEM, V268, P4625
[9]  
STRADER CD, 1988, J BIOL CHEM, V263, P10267
[10]   IDENTIFICATION OF RESIDUES REQUIRED FOR LIGAND-BINDING TO THE BETA-ADRENERGIC-RECEPTOR [J].
STRADER, CD ;
SIGAL, IS ;
REGISTER, RB ;
CANDELORE, MR ;
RANDS, E ;
DIXON, RAF .
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 1987, 84 (13) :4384-4388