An efficient synthesis of some new bisbenzimidazoles via microwave technique

被引:8
作者
Kahveci, Bahittin [1 ]
Karaali, Nesrin [2 ]
Yilmaz, Fatih [2 ]
Mentese, Emre [2 ]
机构
[1] Karadeniz Tech Univ, Dept Nutr & Dietet, Trabzon, Turkey
[2] Recep Tayyip Erdogan Univ, Dept Chem, Rize, Turkey
关键词
Bisbenzimidazole; bisiminoester hydrochloride; microwave synthesis; hydrazine hydrate; ANTIMICROBIAL ACTIVITY; BENZIMIDAZOLE; 2-PHENYLBENZIMIDAZOLE; DERIVATIVES;
D O I
10.3906/kim-1305-17
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
2,2'-[1,4 (1,3)-Phenylenedi(methylene)]bis-1H-benzimidazole derivatives were obtained from the reaction of 1,4- or (1,3)-bisiminoester hydrochloride and o-phenylenediamine derivatives under microwave irradiation. Ester and hydrazide derivatives were prepared from a free NH group. This practical method revealed good results for yield, reaction time, and quick isolation of products.
引用
收藏
页码:423 / 429
页数:7
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