Synthesis and biological activity of dimeric HIV-1 integrase inhibitory peptides

被引：0
作者：
Krajewski, Krzysztof [1 ]
Long, Ya-Qiu [1 ]
Marchand, Christophe [1 ]
Pommier, Yves [1 ]
Roller, Peter P. [1 ]
机构：
[1] NCI, Med Chem Lab, NIH, Frederick, MD 21702 USA
来源：
PEPTIDE REVOLUTION: GENOMICS, PROTEOMICS & THERAPEUTICS | 2004年
关键词：
D O I：
暂无
中图分类号：
Q5 [生物化学]; Q7 [分子生物学];
学科分类号：
071010 ; 081704 ;
摘要：
引用
收藏
页码：329 / 330
页数：2
相关论文
共 50 条
  • [21] Linker-modified quinoline derivatives targeting HIV-1 integrase:: synthesis and biological activity
    Bernard, C
    Zouhiri, F
    Normand-Bayle, M
    Danet, M
    Desmaële, D
    Leh, H
    Mouscadet, JF
    Mbemba, G
    Thomas, CM
    Bonnenfant, S
    Le Bret, M
    d'Angelo, J
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (10) : 2473 - 2476
  • [22] Synthesis and biological evaluation of geminal disulfones as HIV-1 integrase inhibitors
    Meadows, DC
    Mathews, TB
    North, TW
    Hadd, MJ
    Kuo, CL
    Neamati, N
    Gervay-Hague, J
    [J]. JOURNAL OF MEDICINAL CHEMISTRY, 2005, 48 (14) : 4526 - 4534
  • [23] Synthesis and Biological Activities of Quinoline Derivatives as HIV-1 Integrase Inhibitors
    Luo Zai-gang
    Zeng Cheng-chu
    Wang Fang
    He Hong-qiu
    Wang Cun-xin
    Du Hong-guang
    Hu Li-ming
    [J]. CHEMICAL RESEARCH IN CHINESE UNIVERSITIES, 2009, 25 (06) : 841 - 845
  • [24] Synthesis and Biological Activities of Quinoline Derivatives as HIV-1 Integrase Inhibitors
    LUO Zai-gang1
    2. College of Science
    [J]. Chemical Research in Chinese Universities, 2009, 25 (06) : 841 - 845
  • [25] A novel aspochalasin with HIV-1 integrase inhibitory activity from Aspergillus flavipes
    Rochfort, S
    Ford, J
    Ovenden, S
    Wan, SS
    George, S
    Wildman, H
    Tait, RM
    Meurer-Grimes, B
    Cox, S
    Coates, J
    Rhodes, D
    [J]. JOURNAL OF ANTIBIOTICS, 2005, 58 (04) : 279 - 283
  • [26] A Novel Aspochalasin with HIV-1 Integrase Inhibitory Activity from Aspergillus flavipes
    Simone Rochfort
    Joanne Ford
    Simon Ovenden
    Soo San Wan
    Samantha George
    Howard Wildman
    R Murray Tait
    Barbara Meurer-Grimes
    Susan Cox
    Jonathan Coates
    David Rhodes
    [J]. The Journal of Antibiotics, 2005, 58 : 279 - 283
  • [27] Chemical and enzymatic modifications of integric acid and HIV-1 integrase inhibitory activity
    Singh, SB
    Felock, P
    Hazuda, DJ
    [J]. BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2000, 10 (03) : 235 - 238
  • [28] HIV-1 protease and HIV-1 integrase inhibitory substances from Eclipta prostrata
    Tewtrakul, Supinya
    Subhadhirasakul, Sanan
    Cheenpracha, Sarot
    Karalai, Chatchanok
    [J]. PHYTOTHERAPY RESEARCH, 2007, 21 (11) : 1092 - 1095
  • [29] HIV-1 integrase inhibition by dimeric bisbenzimidazoles with different spacer structures
    S. P. Korolev
    V. N. Tashlitsky
    M. A. Smolov
    A. V. Gromyko
    A. L. Zhuze
    Yu. Yu. Agapkina
    M. B. Gottikh
    [J]. Molecular Biology, 2010, 44 : 633 - 641
  • [30] HIV-1 integrase inhibition by dimeric bisbenzimidazoles with different spacer structures
    Korolev, S. P.
    Tashlitsky, V. N.
    Smolov, M. A.
    Gromyko, A. V.
    Zhuze, A. L.
    Agapkina, Yu. Yu.
    Gottikh, M. B.
    [J]. MOLECULAR BIOLOGY, 2010, 44 (04) : 633 - 641
12345