共 94 条
Pregnane X receptor: a double-edged sword
被引:2
作者:

Fang Dao-kui
论文数: 0 引用数: 0
h-index: 0
机构:
Shenzhen Ctr Dis Control & Prevent, Persistent Organ Pollutant Lab, Shenzhen 518020, Guangdong, Peoples R China Shenzhen Ctr Dis Control & Prevent, Persistent Organ Pollutant Lab, Shenzhen 518020, Guangdong, Peoples R China

Zhang Jian-qing
论文数: 0 引用数: 0
h-index: 0
机构:
Shenzhen Ctr Dis Control & Prevent, Persistent Organ Pollutant Lab, Shenzhen 518020, Guangdong, Peoples R China Shenzhen Ctr Dis Control & Prevent, Persistent Organ Pollutant Lab, Shenzhen 518020, Guangdong, Peoples R China
机构:
[1] Shenzhen Ctr Dis Control & Prevent, Persistent Organ Pollutant Lab, Shenzhen 518020, Guangdong, Peoples R China
基金:
中国国家自然科学基金;
关键词:
pregnane X receptor;
protein structure;
function;
CONSTITUTIVE ANDROSTANE RECEPTOR;
DRUG-INDUCED OSTEOMALACIA;
ORPHAN NUCLEAR RECEPTOR;
NF-KAPPA-B;
INFLAMMATORY-BOWEL-DISEASE;
HUMAN CYTOCHROME-P450 3A4;
PRIMARY HUMAN HEPATOCYTES;
CYP3A GENE-EXPRESSION;
XENOBIOTIC RECEPTOR;
CRYSTAL-STRUCTURE;
D O I:
10.3760/cma.j.issn.0366-6999.2009.11.018
中图分类号:
R5 [内科学];
学科分类号:
1002 ;
100201 ;
摘要:
[No abstract available]
引用
收藏
页码:1333 / 1341
页数:9
相关论文
共 94 条
[81]
Coactivator binding promotes the specific interaction between ligand and the pregnane X receptor
[J].
Watkins, RE
;
Davis-Searles, PR
;
Lambert, MH
;
Redinbo, MR
.
JOURNAL OF MOLECULAR BIOLOGY,
2003, 331 (04)
:815-828

Watkins, RE
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Davis-Searles, PR
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Lambert, MH
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Redinbo, MR
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA
[82]
2.1 Å crystal structure of human PXR in complex with the St. John's wort compound hyperforin
[J].
Watkins, RE
;
Maglich, JM
;
Moore, LB
;
Wisely, GB
;
Noble, SM
;
Davis-Searles, PR
;
Lambert, MH
;
Kliewer, SA
;
Redinbo, MR
.
BIOCHEMISTRY,
2003, 42 (06)
:1430-1438

Watkins, RE
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Maglich, JM
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Moore, LB
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Wisely, GB
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Noble, SM
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Davis-Searles, PR
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Lambert, MH
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Kliewer, SA
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Redinbo, MR
论文数: 0 引用数: 0
h-index: 0
机构:
Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA
[83]
Drug therapy - Drug metabolism and variability among patients in drug response
[J].
Wilkinson, GR
.
NEW ENGLAND JOURNAL OF MEDICINE,
2005, 352 (21)
:2211-2221

Wilkinson, GR
论文数: 0 引用数: 0
h-index: 0
机构:
Vanderbilt Univ, Dept Pharmacol, Nashville, TN 37232 USA Vanderbilt Univ, Dept Pharmacol, Nashville, TN 37232 USA
[84]
Lithocholic acid induction of the FGF19 promoter in intestinal cells is mediated by PXR
[J].
Wistuba, Wolfgang
;
Gnewuch, Carsten
;
Liebisch, Gerhard
;
Schmitz, Gerd
;
Langmann, Thomas
.
WORLD JOURNAL OF GASTROENTEROLOGY,
2007, 13 (31)
:4230-4235

Wistuba, Wolfgang
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany

Gnewuch, Carsten
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany

Liebisch, Gerhard
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany

Schmitz, Gerd
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany

Langmann, Thomas
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany Univ Regensburg, Inst Clin Chem & Lab Med, D-93053 Regensburg, Germany
[85]
The impact of pregnane X receptor activation on liver fibrosis
[J].
Wright, M. C.
.
BIOCHEMICAL SOCIETY TRANSACTIONS,
2006, 34
:1119-1123

Wright, M. C.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Newcastle, Sch Clin & Lab Sci, Sch Med, Liver Res Fac Grp, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Univ Newcastle, Sch Clin & Lab Sci, Sch Med, Liver Res Fac Grp, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England
[86]
An essential role for nuclear receptors SXR/PXR in detoxification of cholestatic bile acids
[J].
Xie, W
;
Radominska-Pandya, A
;
Shi, YH
;
Simon, CM
;
Nelson, MC
;
Ong, ES
;
Waxman, DJ
;
Evans, RM
.
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA,
2001, 98 (06)
:3375-3380

Xie, W
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA

Radominska-Pandya, A
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA

Shi, YH
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA

Simon, CM
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA

Nelson, MC
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA

Ong, ES
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA

Waxman, DJ
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA

Evans, RM
论文数: 0 引用数: 0
h-index: 0
机构: Salk Inst Biol Studies, Gene Express Lab, La Jolla, CA 92037 USA
[87]
Intestinal and hepatic CYP3A4 catalyze hydroxylation of 1α,25-dihydroxyvitamin D3:: Implications for drug-induced osteomalacia
[J].
Xu, Y
;
Hashizume, T
;
Shuhart, MC
;
Davis, CL
;
Nelson, WL
;
Sakaki, T
;
Kalhorn, TF
;
Watkins, PB
;
Schuetz, EG
;
Thummel, KE
.
MOLECULAR PHARMACOLOGY,
2006, 69 (01)
:56-65

Xu, Y
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Hashizume, T
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Shuhart, MC
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Davis, CL
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Nelson, WL
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Sakaki, T
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Kalhorn, TF
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Watkins, PB
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Schuetz, EG
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA

Thummel, KE
论文数: 0 引用数: 0
h-index: 0
机构: Univ Washington, Dept Pharmaceut, Seattle, WA 98195 USA
[88]
Crystal structure of the pregnane X receptor-estradiol complex provides insights into endobiotic recognition
[J].
Xue, Yu
;
Moore, Linda B.
;
Orans, Jillian
;
Peng, Li
;
Bencharit, Sompop
;
Kliewer, Steven A.
;
Redinbo, Matthew R.
.
MOLECULAR ENDOCRINOLOGY,
2007, 21 (05)
:1028-1038

Xue, Yu
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Moore, Linda B.
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Orans, Jillian
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Peng, Li
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Bencharit, Sompop
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Kliewer, Steven A.
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA

Redinbo, Matthew R.
论文数: 0 引用数: 0
h-index: 0
机构: Univ N Carolina, Dept Chem, Chapel Hill, NC 27599 USA
[89]
Identification of Ginkgo biloba as a Novel Activator of Pregnane X Receptor
[J].
Yeung, Eugene Y. H.
;
Sueyoshi, Tatsuya
;
Negishi, Masahiko
;
Chang, Thomas K. H.
.
DRUG METABOLISM AND DISPOSITION,
2008, 36 (11)
:2270-2276

Yeung, Eugene Y. H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ British Columbia, Fac Pharmaceut Sci, Vancouver, BC V6T 1Z3, Canada Univ British Columbia, Fac Pharmaceut Sci, Vancouver, BC V6T 1Z3, Canada

Sueyoshi, Tatsuya
论文数: 0 引用数: 0
h-index: 0
机构:
Natl Inst Environm Hlth Sci, NIH, Pharmacogenet Sect, Reprod & Dev Toxicol Lab, Res Triangle Pk, NC USA Univ British Columbia, Fac Pharmaceut Sci, Vancouver, BC V6T 1Z3, Canada

Negishi, Masahiko
论文数: 0 引用数: 0
h-index: 0
机构:
Natl Inst Environm Hlth Sci, NIH, Pharmacogenet Sect, Reprod & Dev Toxicol Lab, Res Triangle Pk, NC USA Univ British Columbia, Fac Pharmaceut Sci, Vancouver, BC V6T 1Z3, Canada

Chang, Thomas K. H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ British Columbia, Fac Pharmaceut Sci, Vancouver, BC V6T 1Z3, Canada Univ British Columbia, Fac Pharmaceut Sci, Vancouver, BC V6T 1Z3, Canada
[90]
Potential role for human cytochrome P450 3A4 in estradiol homeostasis
[J].
Yu, AM
;
Fukamachi, K
;
Krausz, KW
;
Cheung, C
;
Gonzalez, FJ
.
ENDOCRINOLOGY,
2005, 146 (07)
:2911-2919

Yu, AM
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Lab Metab, NIH, Bethesda, MD 20892 USA

Fukamachi, K
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Lab Metab, NIH, Bethesda, MD 20892 USA

Krausz, KW
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Lab Metab, NIH, Bethesda, MD 20892 USA

Cheung, C
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Lab Metab, NIH, Bethesda, MD 20892 USA

Gonzalez, FJ
论文数: 0 引用数: 0
h-index: 0
机构: NCI, Lab Metab, NIH, Bethesda, MD 20892 USA