共 12 条
[1]
Mining a Cathepsin Inhibitor Library for New Antiparasitic Drug Leads
[J].
Ang, Kenny K. H.
;
Ratnam, Joseline
;
Gut, Jiri
;
Legac, Jennifer
;
Hansell, Elizabeth
;
Mackey, Zachary B.
;
Skrzypczynska, Katarzyna M.
;
Debnath, Anjan
;
Engel, Juan C.
;
Rosenthal, Philip J.
;
McKerrow, James H.
;
Arkin, Michelle R.
;
Renslo, Adam R.
.
PLOS NEGLECTED TROPICAL DISEASES,
2011, 5 (05)

Ang, Kenny K. H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Ratnam, Joseline
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Gut, Jiri
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, San Francisco Gen Hosp, Dept Med, San Francisco, CA USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Legac, Jennifer
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, San Francisco Gen Hosp, Dept Med, San Francisco, CA USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Hansell, Elizabeth
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Sandler Ctr Drug Discovery, San Francisco, CA 94143 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Mackey, Zachary B.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Sandler Ctr Drug Discovery, San Francisco, CA 94143 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Skrzypczynska, Katarzyna M.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Sandler Ctr Drug Discovery, San Francisco, CA 94143 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Debnath, Anjan
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Sandler Ctr Drug Discovery, San Francisco, CA 94143 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Engel, Juan C.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Sandler Ctr Drug Discovery, San Francisco, CA 94143 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Rosenthal, Philip J.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, San Francisco Gen Hosp, Dept Med, San Francisco, CA USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

McKerrow, James H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Sandler Ctr Drug Discovery, San Francisco, CA 94143 USA
Univ Calif San Francisco, Dept Pathol, San Francisco, CA 94140 USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Arkin, Michelle R.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA

Renslo, Adam R.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA USA Univ Calif San Francisco, Small Mol Discovery Ctr, San Francisco, CA 94143 USA
[2]
Beaulieu C, 2008, BIOORGAN MED CHEM, V20, P7444
[3]
Falcipain Inhibitors: Optimization Studies of the 2-Pyrimidinecarbonitrile Lead Series
[J].
Coteron, Jose M.
;
Catterick, David
;
Castro, Julia
;
Chaparro, Maria J.
;
Diaz, Beatriz
;
Fernandez, Esther
;
Ferrer, Santiago
;
Gamo, Francisco J.
;
Gordo, Mariola
;
Gut, Jiri
;
de las Heras, Laura
;
Legac, Jennifer
;
Marco, Maria
;
Miguel, Juan
;
Munoz, Vicente
;
Porras, Esther
;
de la Rosa, Juan C.
;
Ruiz, Jose R.
;
Sandoval, Elena
;
Ventosa, Pilar
;
Rosenthal, Philip J.
;
Fiandor, Jose M.
.
JOURNAL OF MEDICINAL CHEMISTRY,
2010, 53 (16)
:6129-6152

Coteron, Jose M.
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Catterick, David
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Synthet Chem, Tonbridge TN11 9AN, Kent, England Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Castro, Julia
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Chaparro, Maria J.
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Diaz, Beatriz
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Fernandez, Esther
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Ferrer, Santiago
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Biol, DDW, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Gamo, Francisco J.
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Biol, DDW, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Gordo, Mariola
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Gut, Jiri
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

de las Heras, Laura
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Legac, Jennifer
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Marco, Maria
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Miguel, Juan
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Munoz, Vicente
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Porras, Esther
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

de la Rosa, Juan C.
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Ruiz, Jose R.
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Sandoval, Elena
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Ventosa, Pilar
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Rosenthal, Philip J.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA

Fiandor, Jose M.
论文数: 0 引用数: 0
h-index: 0
机构:
GlaxoSmithKline, Dept Drug Discovery Chem, Madrid 28760, Spain Univ Calif San Francisco, Dept Med, San Francisco Gen Hosp, San Francisco, CA 94143 USA
[4]
Peptidomimetic nitriles as selective inhibitors for the malarial cysteine protease falcipain-2
[J].
Ehmke, Veronika
;
Kilchmann, Falco
;
Heindl, Cornelia
;
Cui, Kunqiang
;
Huang, Jin
;
Schirmeister, Tanja
;
Diederich, Francois
.
MEDCHEMCOMM,
2011, 2 (08)
:800-804

Ehmke, Veronika
论文数: 0 引用数: 0
h-index: 0
机构:
ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland

Kilchmann, Falco
论文数: 0 引用数: 0
h-index: 0
机构:
ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland

Heindl, Cornelia
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Wurzburg, Inst Pharm & Food Chem, D-97074 Wurzburg, Germany ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland

Cui, Kunqiang
论文数: 0 引用数: 0
h-index: 0
机构:
E China Univ Sci & Technol, Sch Pharm, Shanghai 200237, Peoples R China ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland

Huang, Jin
论文数: 0 引用数: 0
h-index: 0
机构:
E China Univ Sci & Technol, Sch Pharm, Shanghai 200237, Peoples R China ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland

Schirmeister, Tanja
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Wurzburg, Inst Pharm & Food Chem, D-97074 Wurzburg, Germany ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland

Diederich, Francois
论文数: 0 引用数: 0
h-index: 0
机构:
ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland ETH, Organ Chem Lab, CH-8093 Zurich, Switzerland
[5]
Falcipain-2 Inhibitors
[J].
Ettari, Roberta
;
Bova, Floriana
;
Zappala, Maria
;
Grasso, Silvana
;
Micale, Nicola
.
MEDICINAL RESEARCH REVIEWS,
2010, 30 (01)
:136-167

论文数: 引用数:
h-index:
机构:

Bova, Floriana
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Messina, Dipartimento Farmacochim, I-98168 Messina, Italy Univ Messina, Dipartimento Farmacochim, I-98168 Messina, Italy

Zappala, Maria
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Messina, Dipartimento Farmacochim, I-98168 Messina, Italy Univ Messina, Dipartimento Farmacochim, I-98168 Messina, Italy

论文数: 引用数:
h-index:
机构:

论文数: 引用数:
h-index:
机构:
[6]
The discovery of odanacatib (MK-0822), a selective inhibitor of cathepsin K
[J].
Gauthier, Jacques Yves
;
Chauret, Nathalie
;
Cromlish, Wanda
;
Desmarais, Sylvie
;
Duong, Le T.
;
Falgueyret, Jean-Pierre
;
Kimmel, Donald B.
;
Lamontagne, Sonia
;
Leger, Serge
;
LeRiche, Tammy
;
Li, Chun Sing
;
Masse, Frederic
;
Mckay, Daniel J.
;
Nicoll-Griffith, Deborah A.
;
Oballa, Renata A.
;
Palmer, James T.
;
Percival, M. David
;
Riendeau, Denis
;
Robichaud, Joel
;
Rodan, Gideon A.
;
Rodan, Sevgi B.
;
Seto, Carmai
;
Therien, Michel
;
Truong, Vouy-Linh
;
Venuti, Michael C.
;
Wesolowski, Gregg
;
Young, Robert N.
;
Zamboni, Robert
;
Black, W. Cameron
.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS,
2008, 18 (03)
:923-928

Gauthier, Jacques Yves
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Chauret, Nathalie
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Cromlish, Wanda
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Desmarais, Sylvie
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Duong, Le T.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Bone Biol & Osteoporosis Res, West Point, PA USA Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Falgueyret, Jean-Pierre
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Kimmel, Donald B.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Bone Biol & Osteoporosis Res, West Point, PA USA Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Lamontagne, Sonia
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Leger, Serge
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

LeRiche, Tammy
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Li, Chun Sing
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Masse, Frederic
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Mckay, Daniel J.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Nicoll-Griffith, Deborah A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Oballa, Renata A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Palmer, James T.
论文数: 0 引用数: 0
h-index: 0
机构: Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Percival, M. David
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Riendeau, Denis
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Robichaud, Joel
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Rodan, Gideon A.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Bone Biol & Osteoporosis Res, West Point, PA USA Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Rodan, Sevgi B.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Bone Biol & Osteoporosis Res, West Point, PA USA Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Seto, Carmai
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Therien, Michel
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Truong, Vouy-Linh
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Venuti, Michael C.
论文数: 0 引用数: 0
h-index: 0
机构:
Celera Genomics Inc, San Francisco, CA 94080 USA Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Wesolowski, Gregg
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Res Labs, Dept Bone Biol & Osteoporosis Res, West Point, PA USA Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Young, Robert N.
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Zamboni, Robert
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada

Black, W. Cameron
论文数: 0 引用数: 0
h-index: 0
机构:
Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada Merck Frosst Ctr Therapeut Res, Kirkland, PQ H9H 3L1, Canada
[7]
Structural and functional characterization of falcipain-2, a hemoglobinase from the malarial parasite Plasmodium falciparum
[J].
Hogg, Tanis
;
Nagarajan, Krishna
;
Herzberg, Saskia
;
Chen, Lili
;
Shen, Xu
;
Jiang, Hualiang
;
Wecke, Maria
;
Blohmke, Christoph
;
Hilgenfeld, Rolf
;
Schmidt, Christian L.
.
JOURNAL OF BIOLOGICAL CHEMISTRY,
2006, 281 (35)
:25425-25437

Hogg, Tanis
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

Nagarajan, Krishna
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

Herzberg, Saskia
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

Chen, Lili
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

Shen, Xu
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

Jiang, Hualiang
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

Wecke, Maria
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

Blohmke, Christoph
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany

论文数: 引用数:
h-index:
机构:

Schmidt, Christian L.
论文数: 0 引用数: 0
h-index: 0
机构: Med Univ Lubeck, Inst Biochem, Ctr Struct & Cell Biol Med, D-23538 Lubeck, Germany
[8]
Structures of Falcipain-2 and Falcipain-3 Bound to Small Molecule Inhibitors: Implications for Substrate Specificity
[J].
Kerr, Lain D.
;
Lee, Ji H.
;
Pandey, Kailash C.
;
Harrison, Amanda
;
Sajid, Mohammed
;
Rosenthal, Philip J.
;
Brinen, Linda S.
.
JOURNAL OF MEDICINAL CHEMISTRY,
2009, 52 (03)
:852-857

Kerr, Lain D.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Lee, Ji H.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Pandey, Kailash C.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, San Francisco Gen Hosp, Dept Med, San Francisco, CA 94143 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Harrison, Amanda
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, San Francisco Gen Hosp, Dept Med, San Francisco, CA 94143 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Sajid, Mohammed
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Pathol, San Francisco, CA 94158 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Rosenthal, Philip J.
论文数: 0 引用数: 0
h-index: 0
机构: Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA

Brinen, Linda S.
论文数: 0 引用数: 0
h-index: 0
机构:
Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA Univ Calif San Francisco, Dept Mol & Cellular Pharmacol, San Francisco, CA 94158 USA
[9]
Analysis of non-peptidic compounds as potential malarial inhibitors against Plasmodial cysteine proteases via integrated virtual screening workflow
[J].
Musyoka, Thommas M.
;
Kanzi, Aquillah M.
;
Lobb, Kevin A.
;
Bishop, Ozlem Tastan
.
JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS,
2016, 34 (10)
:2084-2101

Musyoka, Thommas M.
论文数: 0 引用数: 0
h-index: 0
机构:
Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa

Kanzi, Aquillah M.
论文数: 0 引用数: 0
h-index: 0
机构:
Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa
Univ Pretoria, FABI, Fac Nat & Agr Sci, Dept Genet, Pretoria, South Africa Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa

Lobb, Kevin A.
论文数: 0 引用数: 0
h-index: 0
机构:
Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa
Rhodes Univ, Dept Chem, POB 94, ZA-6140 Grahamstown, South Africa Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa

Bishop, Ozlem Tastan
论文数: 0 引用数: 0
h-index: 0
机构:
Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa Rhodes Univ, Dept Biochem & Microbiol, Res Unit Bioinformat RUBi, POB 94, ZA-6140 Grahamstown, South Africa
[10]
Discovery of a Selective Series of Inhibitors of Plasmodium falciparum HDACs
[J].
Ontoria, Jesus M.
;
Paonessa, Giacomo
;
Ponzi, Simona
;
Ferrigno, Federica
;
Nizi, Emanuela
;
Biancofiore, Ilaria
;
Malancona, Savina
;
Graziani, Rita
;
Roberts, David
;
Willis, Paul
;
Bresciani, Alberto
;
Gennari, Nadia
;
Cecchetti, Ottavia
;
Monteagudo, Edith
;
Orsale, Maria V.
;
Veneziano, Maria
;
Di Marco, Annalise
;
Cellucci, Antonella
;
Laufer, Ralph
;
Altamura, Sergio
;
Summa, Vincenzo
;
Harper, Steven
.
ACS MEDICINAL CHEMISTRY LETTERS,
2016, 7 (05)
:454-459

Ontoria, Jesus M.
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Paonessa, Giacomo
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Ponzi, Simona
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Ferrigno, Federica
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Nizi, Emanuela
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Biancofiore, Ilaria
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Malancona, Savina
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Graziani, Rita
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Roberts, David
论文数: 0 引用数: 0
h-index: 0
机构:
ICC, Med Malaria Venture, Route Prebois 20,POB 1826, CH-1215 Geneva, Switzerland IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Willis, Paul
论文数: 0 引用数: 0
h-index: 0
机构:
ICC, Med Malaria Venture, Route Prebois 20,POB 1826, CH-1215 Geneva, Switzerland IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Bresciani, Alberto
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Gennari, Nadia
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Cecchetti, Ottavia
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Monteagudo, Edith
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Orsale, Maria V.
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Veneziano, Maria
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Di Marco, Annalise
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Cellucci, Antonella
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Laufer, Ralph
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy
Teva Pharmaceut Ind Ltd, Discovery & Product Dev, POB 8077, IL-4250843 Netanya, Israel IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Altamura, Sergio
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Summa, Vincenzo
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy

Harper, Steven
论文数: 0 引用数: 0
h-index: 0
机构:
IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy
IRBM Sci Pk, Dept Biol, Via Pontina Km 30,600, I-00071 Rome, Italy IRBM Sci Pk, Dept Chem, Via Pontina Km 30,600, I-00071 Rome, Italy