Efficient Synthesis of thieno[2,3-d]pyrimidin-4(4H)-ones by the aza-Wittig Methodology

被引:0
作者
Chen, Hong [1 ]
Yan, Kai [1 ]
Liu, Ming-Guo [1 ]
机构
[1] China Three Gorges Univ, Hubei Key Lab Nat Prod Res & Dev, Yichang, Hubei Prov, Peoples R China
来源
2011 INTERNATIONAL CONFERENCE ON FUZZY SYSTEMS AND NEURAL COMPUTING (FSNC 2011), VOL III | 2011年
关键词
INTRODUCTION; RESULTS AND DISCUSSION; CONCLUSIONS; EXPERIMENTAL SECTION; FACILE SYNTHESIS; DERIVATIVES;
D O I
暂无
中图分类号
TQ [化学工业];
学科分类号
0817 ;
摘要
The carbodiimides 4, obtained from the aza-Wittig reaction of iminophosphorane 3 with aromatic isocyanates' reacted with aliphatic amines or alcohols to give 2-substituted thieno[2,3-d]pyrimidin-4(4H)-ones 6 in the presence of catalytic amount of sodium alkoxide in good yields.
引用
收藏
页码:144 / 147
页数:4
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