Dissolution improvement of high drug-loaded solid dispersion

被引:72
作者
Okonogi, Siriporn [1 ]
Puttipipatkhachorn, Satit
机构
[1] Chiang Mai Univ, Fac Pharm, Dept Pharmaceut Sci, Chiang Mai 50200, Thailand
[2] Mahidol Univ, Fac Pharm, Dept Mfg Pharm, Bangkok 10400, Thailand
关键词
ofloxacin; ternary solid dispersion; polysorbate; 80; dissolution; drug loading;
D O I
10.1208/pt070252
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
This study focused on an investigation of a high drug-loaded solid dispersion system consisting of drug, carrier, and surfactant. Solid dispersions of a water-insoluble ofloxacin (OFX) with polyethylene glycol (PEG) of different molecular weights, namely binary solid dispersion systems, were prepared at drug to carrier not less than 5:5. Polysorbate 80, a nonionic surfactant, was incorporated into the binary solid dispersion systems as the third component to obtain the ternary solid dispersion systems. The powder x-ray diffraction and differential scanning calorimetric studies indicated that crystalline OFX existed in the solid dispersions with high drug loading. However, a decreased crystallinity of the solid dispersions obtained revealed that a portion of OFX was in an amorphous state. The results indicated a remarkably improved dissolution of drug from the ternary solid dispersion systems when compared with the binary solid dispersion systems. This was because of polysorbate 80, which improved wettability and solubilized the non-molecularly dispersed or crystalline fraction of OFX.
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页数:6
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