共 50 条
- [21] GDC-0077 is a selective PI3K alpha inhibitor with robust efficacy in PIK3CA mutant hormone-positive breast cancer modelsCANCER RESEARCH, 2020, 80 (04)Edgar, Kyle论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHong, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASong, Kyung论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASchmidt, Steven论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHafner, Marc论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAArrazate, Alfonso论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWilliams, Erin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADe La Cruz, Cecile论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAOeh, Jason论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASampath, Deepak论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAStaben, Steve论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAFriedman, Lori论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
- [22] Generation of a novel PIK3CA mutated duodenal cancer mouse model and evaluation of PI3K inhibitor therapeutic effectsCANCER SCIENCE, 2024, 115 : 1893 - 1893论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:论文数: 引用数: h-index:机构:Hirotani, Akane论文数: 0 引用数: 0 h-index: 0机构: Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Gastroenterol Ctr, Dept Gastroenterol, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, JapanSawada, Atsushi论文数: 0 引用数: 0 h-index: 0机构: Yokohama City Univ, Med Ctr, Gastroenterol Ctr, Dept Gastroenterol, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, JapanHirasawa, Kingo论文数: 0 引用数: 0 h-index: 0机构: Yokohama City Univ, Med Ctr, Gastroenterol Ctr, Dept Gastroenterol, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, JapanNozaki, Akito论文数: 0 引用数: 0 h-index: 0机构: Yokohama City Univ, Med Ctr, Gastroenterol Ctr, Dept Gastroenterol, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, JapanNumata, Kazushi论文数: 0 引用数: 0 h-index: 0机构: Yokohama City Univ, Med Ctr, Gastroenterol Ctr, Dept Gastroenterol, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, JapanKunisaki, Chikara论文数: 0 引用数: 0 h-index: 0机构: Yokohama City Univ, Dept Surg, Gastroenterol Ctr, Med Ctr, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, JapanMaeda, Shin论文数: 0 引用数: 0 h-index: 0机构: Yokohama City Univ, Dept Gastroenterol, Yokohama, Kanagawa, Japan Yokohama City Univ, Med Ctr, Div Canc Genome Med, Yokohama, Kanagawa, Japan
- [23] Effect of combined treatment with a pan-PI3K inhibitor or an isoform-specific PI3K inhibitor and everolimus on cell proliferation in GH-secreting pituitary tumour in an experimental settingENDOCRINE, 2018, 62 (03) : 663 - 680Pivonello, Claudia论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyPatalano, Roberta论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalySolari, Domenico论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Neurosci, Div Neurochirurg Sci Riprod & Odontostomatol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyAuriemma, Renata S.论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyFrio, Federico论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Neurosci, Div Neurochirurg Sci Riprod & Odontostomatol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyVitulli, Francesca论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Neurosci, Div Neurochirurg Sci Riprod & Odontostomatol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyGrasso, Ludovica F. S.论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyDi Cera, Marialuisa论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyDe Martino, Maria Cristina论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyCavallo, Luigi M.论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Neurosci, Div Neurochirurg Sci Riprod & Odontostomatol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyCappabianca, Paolo论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Neurosci, Div Neurochirurg Sci Riprod & Odontostomatol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyColao, Annamaria论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, ItalyPivonello, Rosario论文数: 0 引用数: 0 h-index: 0机构: Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy Dipartimento Med Clin & Chirurg, Sez Endocrinol, Naples, Italy
- [24] Discovery of GDC-0032: A beta-sparing PI3K inhibitor active against PIK3CA mutant tumors.CANCER RESEARCH, 2013, 73 (08)Olivero, Alan G.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHeffron, Timothy P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABaumgardner, Matthew论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABelvin, Marcia论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USARoss, Leanne Berry论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABlaquiere, Nicole论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USABradley, Erin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USACastanedo, Georgette论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADerynck, Mika论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADo, Steven论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADotson, Jennafer论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USADudley, Danette论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAEdgar, Kyle论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAFolkes, Adrian论文数: 0 引用数: 0 h-index: 0机构: Piramed Pharma, Slough, Berks, England Genentech Inc, San Francisco, CA 94080 USAFrancis, Ross论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAGianetti, Tony论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAGoldsmith, Richard论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAGoldsmith, Paul论文数: 0 引用数: 0 h-index: 0机构: Piramed Pharma, Slough, Berks, England Genentech Inc, San Francisco, CA 94080 USAGuan, Jane论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAHarrison, Trevor论文数: 0 引用数: 0 h-index: 0机构: Argenta Discovery, Harlow, Essex, England Genentech Inc, San Francisco, CA 94080 USAHeald, Robert论文数: 0 引用数: 0 h-index: 0机构: Argenta Discovery, Harlow, Essex, England Genentech Inc, San Francisco, CA 94080 USAHsu, Jerry论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAJackson, Phillip论文数: 0 引用数: 0 h-index: 0机构: Argenta Discovery, Harlow, Essex, England Genentech Inc, San Francisco, CA 94080 USAJones, Graham论文数: 0 引用数: 0 h-index: 0机构: Argenta Discovery, Harlow, Essex, England Genentech Inc, San Francisco, CA 94080 USAKim, Amy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAKolesnikov, Aleks论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALackner, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALee, Leslie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALesnick, John论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USALewis, Cristina论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAMamounas, Michael论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAMcLean, Neville论文数: 0 引用数: 0 h-index: 0机构: Argenta Discovery, Harlow, Essex, England Genentech Inc, San Francisco, CA 94080 USAMurray, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USANdubaku, Chudi论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USANonomiya, Jim论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAPang, Jodie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAPegg, Neil论文数: 0 引用数: 0 h-index: 0机构: Piramed Pharma, Slough, Berks, England Genentech Inc, San Francisco, CA 94080 USAPrior, Wei Wei论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASalphati, Laurent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASampath, Deepack论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASideris, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASiu, Michael论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAStaben, Steven论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USASutherlin, Daniel论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAUltsch, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWallin, Jeff论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWang, Lan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAWiesmann, Christian论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAZhang, Xiaolin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USAFriedman, Lori S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
- [25] Phase I study of BYL719, an alpha-specific PI3K inhibitor, in patients with PIK3CA mutant advanced solid tumors: preliminary efficacy and safety in patients with PIK3CA mutant ER -positive (ER plus ) metastatic breast cancer (MBC)CANCER RESEARCH, 2012, 72Juric, D.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USAArgiles, G.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USABurns, H. A.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USAGonzalez-Angulo, A. M.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USASaura, C.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USAQuadt, C.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USADouglas, M.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USADemanse, D.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USADe Buck, S.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USABaselga, J.论文数: 0 引用数: 0 h-index: 0机构: Massachussetts Gen Hosp, Ctr Canc, Boston, MA USA
- [26] Gedatolisib, a pan-PI3K/mTOR inhibitor, shows superior potency and efficacy relative to other PI3K/AKT/mTOR pathway inhibitors in breast cancer modelsCANCER RESEARCH, 2024, 84 (09)Rossetti, Stefano论文数: 0 引用数: 0 h-index: 0Broege, Aaron论文数: 0 引用数: 0 h-index: 0Sen, Adrish论文数: 0 引用数: 0 h-index: 0Khan, Salmaan论文数: 0 引用数: 0 h-index: 0MacNeil, Ian论文数: 0 引用数: 0 h-index: 0Molden, Jhomary论文数: 0 引用数: 0 h-index: 0Gorbatchevsky, Igor论文数: 0 引用数: 0 h-index: 0Sullivan, Brian F.论文数: 0 引用数: 0 h-index: 0Laing, Lance论文数: 0 引用数: 0 h-index: 0
- [27] Which Is the Most Appropriate PI3K Inhibitor for Breast Cancer Patients with or without PIK3CA Status Mutant? A Systematic Review and Network Meta-AnalysisBIOMED RESEARCH INTERNATIONAL, 2020, 2020Wang, Shu论文数: 0 引用数: 0 h-index: 0机构: China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R ChinaLiu, Mingyue论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Clin Pharm, Shenyang 110016, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R ChinaLian, Siheng论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Clin Pharm, Shenyang 110016, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R ChinaLiu, Naiming论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Clin Pharm, Shenyang 110016, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R ChinaZhang, Guibin论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Clin Pharm, Shenyang 110016, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R ChinaZhao, Qingchun论文数: 0 引用数: 0 h-index: 0机构: China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R China Shenyang Pharmaceut Univ, Dept Clin Pharm, Shenyang 110016, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R ChinaZhang, Yingshi论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Dept Clin Pharm, Shenyang 110016, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R ChinaJian, Lingyan论文数: 0 引用数: 0 h-index: 0机构: China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R China China Med Univ, Shengjing Hosp, Dept Pharm, Shenyang 110004, Peoples R China
- [28] The AKT inhibitor AZD5363 is selectively active in PIK3CA mutant gastric cancer cell lines, and sensitizes a gastric cancer explant model to docetaxelCANCER RESEARCH, 2012, 72Li, Jing论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaDavies, Barry R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Macclesfield, Cheshire, England AstraZeneca, Shanghai, Peoples R ChinaZhou, Minhua论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaZhang, Jingchuan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaXu, Yan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaTang, Lili论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaWang, Huiying论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaLiu, Charles论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaYin, Xiaolu论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaJi, Qunsheng论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R ChinaYu, Derek Dehua论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Shanghai, Peoples R China AstraZeneca, Shanghai, Peoples R China
- [29] PRECLINICAL DEVELOPMENT OF THE PI3K ALPHA SELECTIVE AND PIK3CA MUTANT SELECTIVE INHIBITOR GDC-0077 AND PREDICTION OF ITS HUMAN PHARMACOKINETICSDRUG METABOLISM AND PHARMACOKINETICS, 2019, 34 (01) : S37 - S37Pang, Jodie论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USABaumgardner, Matthew论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USABraun, Marie-Gabrielle论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USACheong, Jonathan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAEdgar, Kyle论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAFriedman, Lori论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAHanan, Emily论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAJaochico, Allan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAMa, Shuguang论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAPlise, Emile论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USASchmidt, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USALiu, Ning论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USASong, Kyung论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USAStaben, Steve论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USASalphati, Laurent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Genentech Inc, San Francisco, CA USA
- [30] Gedatolisib, a well-tolerated pan-PI3K/mTOR inhibitor, exhibits potent therapeutic effects on endometrial cancer models regardless of their PI3K pathway mutational statusCANCER RESEARCH, 2023, 83 (07)Rossetti, Stefano论文数: 0 引用数: 0 h-index: 0Broege, Aaron论文数: 0 引用数: 0 h-index: 0MacNeil, Ian论文数: 0 引用数: 0 h-index: 0Rich, Ben论文数: 0 引用数: 0 h-index: 0Molden, Jhomary论文数: 0 引用数: 0 h-index: 0Sullivan, Brian论文数: 0 引用数: 0 h-index: 0Laing, Lance论文数: 0 引用数: 0 h-index: 0