One-pot synthesis of pyrimidines under solvent-free conditions

被引：13

作者：

Ghorbani-Vaghei, Ramin ^{[1
]}

Karimi-Nami, Rahman ^{[2
]}

Toghraei-Semiromi, Zahra ^{[1
]}

Amiri, Mostafa ^{[1
]}

Salimi, Zahra ^{[1
]}

Ghavidel, Mehdi ^{[3
]}

机构：

[1] Bu Ali Sina Univ, Fac Chem, Dept Organ Chem, Hamadan 65174, Iran

[2] Univ Tehran, Sch Chem, Univ Coll Sci, Tehran, Iran

[3] Urmia Univ, Dept Chem, Orumiyeh 57154, Iran

来源：

COMPTES RENDUS CHIMIE | 2014年 / 17卷 / 04期

关键词：

Pyrimidine; Multicomponent reaction; Triethoxymethane; Ammonium acetate; Solvent-free; TBBDA; DERIVATIVES; CHEMISTRY; REAGENTS; MILD;

D O I：

10.1016/j.crci.2013.07.010

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

N,N,N',N'-Tetrabromobenzene-1,3-disulfonamide was used as an efficient catalyst for the one-pot synthesis of pyrimidine derivatives in excellent yields from triethoxymethane, ammonium acetate, and various ketone derivatives at 100-110 degrees C under solvent-free conditions. (C) 2013 Academie des sciences. Published by Elsevier Masson SAS. All rights reserved.

引用

页码：324 / 330

页数：7

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