NaIO4-Catalyzed One-Pot Synthesis of Dihydropyrimidinones at Room Temperature under Solvent-Free Conditions

被引：23

作者：

Jing, X. ^{[1
]}

Li, Z. ^{[1
]}

Pan, X. ^{[1
]}

Shi, Y. ^{[1
]}

Yan, C. ^{[1
]}

机构：

[1] Yangzhou Univ, Coll Chem & Chem Engn, Yangzhou 225002, Peoples R China

来源：

JOURNAL OF THE IRANIAN CHEMICAL SOCIETY | 2009年 / 6卷 / 03期

基金：

中国国家自然科学基金;

关键词：

Pyrimidinones; Sodium periodate; Biginelli reaction; Solvent-free conditions; BIGINELLI; PROTOCOL;

D O I：

10.1007/BF03246529

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

Sodium periodate efficiently catalyzed the three-component Biginelli reaction of an aldehyde, alpha beta-keto ester or beta-keto ketone, and urea or thiourea at room temperature under solvent-free conditions and afforded the corresponding 3,4-dihydropyrimidine-2-(1H)-ones in excellent yields.

引用

页码：514 / 518

页数：5

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