Rearrangement of pyrrolo[2,1-c][1,4]benzodiazepines into cyclopenta[b][1,4]benzodiazepines under microwave or conventional heating conditions.

被引：18

作者：

Gillard, AC ^{[1
]}

Fabis, F ^{[1
]}

JolivetFouchet, S ^{[1
]}

Rault, S ^{[1
]}

机构：

[1] UNIV CAEN,UFR SCI PHARMACEUT,CTR ETUD & RECH MEDICAMENT NORMANDIE,F-14032 CAEN,FRANCE

来源：

TETRAHEDRON LETTERS | 1997年 / 38卷 / 13期

关键词：

D O I：

10.1016/S0040-4039(97)00359-6

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Microwave or conventional heating of 2-hydroxy or 2-oxo-pyrrolo[2,1-c][1,4]benzodiazepinediones in boiling phosphoryl chloride led to cyclopenta[b][1,4]benzodiazepines. (C) 1997 Published by Elsevier Science Ltd.

引用

页码：2271 / 2274

页数：4

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