Synthesis of 3-ferrocenyl-3,3a,4,5-tetrahydro-2H-benzo[g]indazoles

被引：0
|
作者：
Klimova, E
Klimova, T
Apan, TR
Camacho, AN
Esparza, RM
Zea, CD
García, MM
机构：
[1] Univ Nacl Autonoma Mexico, Fac Chem, Mexico City 04510, DF, Mexico
[2] Univ Nacl Autonoma Mexico, Inst Chem, Mexico City 04510, DF, Mexico
来源：
HETEROCYCLES | 2004年 / 63卷 / 05期
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The reactions of E-2-ferrocenylmethylidenetetralones with hydrazine proceed diastereoselectively, forming the cis isomers of diazatricycles in high yields. The studies of the anti-inflammatory activity of E-2-ferrocenylmethylidenetetralones and N-acetylindazoles showed a moderate activity in a TPA model. The structure of 2-acetyl-3-ferrocenyl-6-methoxy-3,3a,4,5-tetrahydro-2H-benzo[g]indazole was confirmed by X-Ray diffraction analysis.
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页码：1045 / 1056
页数：12
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