Synthesis and antifungal activity of some new 1-aryl/heteroaryl-4-methyl-1,2,4-triazolo [4,3-a] quinoxalines

被引：0

作者：

Aggarwal, Ranjana ^{[1
]}

Sumran, Garima

Kumar, Rajiv

Aggarwal, Ashok

Parkash, Vipin

机构：

[1] Kurukshetra Univ, Dept Chem, Kurukshetra 136119, Haryana, India

[2] Kurukshetra Univ, Dept Bot, Kurukshetra 136119, Haryana, India

来源：

INDIAN JOURNAL OF HETEROCYCLIC CHEMISTRY | 2006年 / 16卷 / 01期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A simple and highly efficient synthesis of some 1-aryl/heteroaryl-4-methyl-1,2,4-triazolo [4,3-a] quinoxalines (3) by oxidative cyclization of arene carbaldehyde-3-methylquinoxalin-2-yl hydrazones (2) with iodobenzene diacetate (IBD) in dichloromethane is described. Some of the compounds were tested in vitro for their antifungal activity against Fusarium udum, Helminthosporium sp. and Aspergillus flavus.

引用

页码：1 / 4

页数：4

共 17 条

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