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- [1] Structure-Based Design of Novel Inhibitors of the MDM2-p53 InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2012, 55 (11) : 4936 - 4954Rew, Yosup论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USADe Turiso, Felix Gonzalez-Lopez论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USABartberger, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USABeck, Hilary P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USACanon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAChen, Ada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAChow, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USADeignan, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAFox, Brian M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAGustin, Darin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAJiang, Min论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAJiao, Xianyun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAJin, Lixia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAKayser, Frank论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAKopecky, David J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USALi, Yihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USALo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USALong, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAMichelsen, Klaus论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAOliner, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAOsgood, Tao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USARagains, Mark论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmaceut, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USASaiki, Anne Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USASchneider, Steve论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAToteva, Maria论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmaceut, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAYakowec, Peter论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAYan, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAYu, Dongyin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAZhou, Jing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAMedina, Julio C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USAOlson, Steven H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Dept Therapeut Discovery, San Francisco, CA 94080 USA
- [2] Discovery of AM-8553: Structure-based design of novel piperidinone inhibitors of the MDM2-p53 interactionABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 244Rew, Yosup论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USASun, Daqing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USADe Turiso, Felix Gonzalez Lopez论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USABartberger, Michael D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USABeck, Hilary P.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USACanon, Jude论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAChen, Ada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAChow, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USADeignan, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAFox, Brian M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAGustin, Darin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAHuang, Xin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAJiang, Min论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAJiao, Xianyun论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAJin, Lixia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAKayser, Frank论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAKopecky, David J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USALi, Yihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USALo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USALong, Alexander M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAMichelsen, Klaus论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, Thousand Oaks, CA 91320 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAOliner, Jonathan D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAOsgood, Tao论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USARagains, Mark论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmaceut, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USASaiki, Anne Y.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USASchneider, Steve论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAToteva, Maria论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmaceut, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAYakowec, Peter论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, Cambridge, MA 02142 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAYan, Xuelei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAYe, Qiuping论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAYu, Dongyin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Oncol Res, Thousand Oaks, CA 91320 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAZhou, Jing论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAMedina, Julio C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USAOlson, Steven H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA Amgen Inc, Therapeut Discovery, San Francisco, CA 94080 USA
- [3] Structure-Based Design of Potent and Orally Active Isoindolinone Inhibitors of MDM2-p53 Protein-Protein InteractionJOURNAL OF MEDICINAL CHEMISTRY, 2021, 64 (07) : 4071 - 4088Chessari, Gianni论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHardcastle, Ian R.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandAhn, Jong Sook论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandAnil, Burcu论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Dept Biochem, Oxford OX1 3QU, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandAnscombe, Elizabeth论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Dept Biochem, Oxford OX1 3QU, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBawn, Ruth H.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBevan, Luke D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBlackburn, Timothy J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandBuck, Ildiko论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCano, Celine论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCarbain, Benoit论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCastro, Juan论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCons, Ben论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandCully, Sarah J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandEndicott, Jane A.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandFazal, Lynsey论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandGolding, Bernard T.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandGriffin, Roger J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHaggerty, Karen论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHarnor, Suzannah J.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHearn, Keisha论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHobson, Stephen论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHolvey, Rhian S.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandHoward, Steven论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandJennings, Claire E.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandJohnson, Christopher N.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, England论文数: 引用数: h-index:机构:Miller, Duncan C.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandNewell, David R.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandNoble, Martin E. M.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandReeks, Judith论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandRevill, Charlotte H.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandRiedinger, Christiane论文数: 0 引用数: 0 h-index: 0机构: Univ Oxford, Dept Biochem, Oxford OX1 3QU, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandSt Denis, Jeffrey D.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandTamanini, Emiliano论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandThomas, Huw论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandThompson, Neil T.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandVinkovic, Mladen论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandWedge, Stephen R.论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandWilliams, Pamela A.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandWilsher, Nicola E.论文数: 0 引用数: 0 h-index: 0机构: Astex Pharmaceut, Cambridge CB4 0QA, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandZhang, Bian论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Sch Nat & Environm Sci, Canc Res UK Newcastle Drug Discovery Unit, Ctr Canc,Chem, Newcastle Upon Tyne NE1 7RU, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, EnglandZhao, Yan论文数: 0 引用数: 0 h-index: 0机构: Newcastle Univ, Fac Med Sci, Canc Res UK Newcastle Drug Discovery Unit, Newcastle Upon Tyne NE2 4HH, Tyne & Wear, England Astex Pharmaceut, Cambridge CB4 0QA, England
- [4] Structure-based design of spiro-oxindoles as potent, specific small-molecule inhibitors of the MDM2-p53 interactionJOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (12) : 3432 - 3435Ding, Ke论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USALu, Yipin论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USANikolovska-Coleska, Zaneta论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAWang, Guoping论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAQiu, Su论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAShangary, Sanjeev论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAGao, Wei论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAQin, Dongguang论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAStuckey, Jeanne论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAKrajewski, Krzysztof论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USARoller, Peter P.论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USAWang, Shaomeng论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Ctr Comprehens Canc, Ann Arbor, MI 48109 USA
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