Synthesis of phthalimido or succinimido[2-aryl-4-oxo-3-{2-phenyl-4(3H)-quinazolinon-3-yl}-1,3-thiazolidin-5-yl]ethanoate

被引：0
|
作者：
Sharma, Shweta [1 ]
Sharma, Chirag [1 ]
Thadhaney, Bhawana [1 ]
Talesara, G. L. [1 ]
机构：
[1] ML Sukhadia Univ, Dept Chem, Synthet Organ Chem Lab, Udaipur 313001, Rajasthan, India
来源：
JOURNAL OF THE INDIAN CHEMICAL SOCIETY | 2009年 / 86卷 / 04期
关键词：
N-Hydroxyphthalimide; N-hydroxysuccinimide; benzoxazine; quinazolinone; thiazolidin; DERIVATIVES; AGENTS;
D O I：
暂无
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
Treatment of benzoxazine I with hydrazine hydrate in ethanol furnished 3-amino-2-phenylquinazolin-4-(3H)-one 2, which upon condensation with aldehydes 3a-d yielded the corresponding 3-arylideneamino derivatives 4a-d. Cyclization of these derivatives using mercaptosuccinic acid afforded 1,3-thiazolidin-4-one ethanoic acids 5a-d, which after esterification with N-hydroxyphthalimide or N-hydroxysuccinimide via acid chlorides produced the respective ethanoic esters 7a-e.
引用
收藏
页码：397 / 401
页数：5
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