Discovery and SAR exploration of a novel series of [1,2,4] triazolo[1,5-a]pyridines as potent and selective RSK inhibitors

被引:0
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作者
Cashion, Dan K. [1 ]
Robinson, Dale [1 ]
Krenitsky, Veronique Plantevin [1 ]
Torres, Eduardo [1 ]
Bahmanyara, Sogole [1 ]
Bates, Robert [2 ]
Delker, Silvia L. [3 ]
Pagarigan, Barbara [3 ]
Fang, Wei [3 ]
Chamberlain, Phil [3 ]
机构
[1] Celgene, Med Chem, San Diego, CA 92121 USA
[2] Celgene, Inflammat Res, San Diego, CA 92121 USA
[3] Celgene, Biochem & Struct Biol, San Diego, CA 92121 USA
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O6 [化学];
学科分类号
0703 ;
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312-MEDI
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页数:1
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